Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 3493
TargetTyrosine-protein kinase JAK3(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(US10011571, Example 23 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 11nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK3(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(US10011571, Example 7 | Preparation of N-(3-(5-chl...)
Affinity DataIC50: 11nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK3(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(US10011571, Example 22 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 21nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 3(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(US10011571, Example 23 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 42nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(US10011571, Example 7 | Preparation of N-(3-(5-chl...)
Affinity DataIC50: 105nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 3(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(US10011571, Example 7 | Preparation of N-(3-(5-chl...)
Affinity DataIC50: 107nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(US10011571, Example 7 | Preparation of N-(3-(5-chl...)
Affinity DataIC50: 162nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(US10011571, Example 23 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 173nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(US10011571, Example 22 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 279nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Blk(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(US10011571, Example 7 | Preparation of N-(3-(5-chl...)
Affinity DataIC50: 286nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(US10011571, Example 7 | Preparation of N-(3-(5-chl...)
Affinity DataIC50: 319nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(US10011571, Example 23 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 664nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 1(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(US10011571, Example 7 | Preparation of N-(3-(5-chl...)
Affinity DataIC50: 698nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Blk(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(US10011571, Example 23 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 855nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 1(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(US10011571, Example 23 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.23E+3nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(US10011571, Example 7 | Preparation of N-(3-(5-chl...)
Affinity DataIC50: 1.40E+3nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Blk(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(US10011571, Example 22 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.66E+3nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(US10011571, Example 23 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.92E+3nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402040(US10011571, Example 7 | Preparation of N-(3-(5-chl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402042(US10011571, Example 23 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetSerine/threonine-protein kinase TBK1(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(US10011571, Example 22 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 1(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(US10011571, Example 22 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 3(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(US10011571, Example 22 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(US10011571, Example 22 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(US10011571, Example 22 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetTyrosine-protein kinase ITK/TSK(Human)
Shenzhen Chipscreen Biosciences

US Patent
LigandPNGBDBM402041(US10011571, Example 22 | Preparation of N-(3-(5-ch...)
Affinity DataIC50: 1.00E+4nMAssay Description:Briefly, according to the requirements of different kinase reactions, 0.2 μL test compound (50 μM, dissolved in dimethyl sulfoxide (DMSO)) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent