Compile Data Set for Download or QSAR
Report error Found 111 Enz. Inhib. hit(s) with all data for entry = 3506
TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402175BDBM402175(US10011607, 9 | (9aS)-7-[2,6-difluoro-4-(2- phenyl...)
Affinity DataEC50:  29nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402282BDBM402282(US10011607, 110 | (9aS)-7-[2,6-difluoro-4-[2-(2- f...)
Affinity DataEC50:  31nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402193BDBM402193(US10011607, 26 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  36nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402194BDBM402194(US10011607, 27 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  39nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402171BDBM402171(US10011607, 5 | (9aS)-7-[2,6-difluoro-4-(2- phenyl...)
Affinity DataEC50:  46nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402200BDBM402200(US10011607, 33 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  46nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402225BDBM402225(US10011607, 54 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  48nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402204BDBM402204(US10011607, 37 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  55nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402217BDBM402217(US10011607, 47 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  55nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402283BDBM402283(US10011607, 111 | (9aS)-7-[2,6-difluoro-4-[2-(2- f...)
Affinity DataEC50:  56nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402281BDBM402281(US10011607, 109 | (9aS)-7-[2,6-difluoro-4-[2-(2- f...)
Affinity DataEC50:  56nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402189BDBM402189(US10011607, 23 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  61nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402277BDBM402277(US10011607, 105 | (9aR)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  61nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402258BDBM402258(US10011607, 86 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  68nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402185BDBM402185(US10011607, 19 | (9aS)-2-(2-chloro-4-pyridyl)- 7-[...)
Affinity DataEC50:  69nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402173BDBM402173(US10011607, 7 | (9aS)-7-[2,6-difluoro-4-(2- phenyl...)
Affinity DataEC50:  73nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402260BDBM402260(US10011607, 88 | (9aRS)-2-[(3-chloro- phenyl)methy...)
Affinity DataEC50:  73nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402187BDBM402187(US10011607, 21 | (9aS)-2-(6-chloro-3-pyridyl)- 7-[...)
Affinity DataEC50:  73nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402211BDBM402211(US10011607, 42 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  73nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402221BDBM402221(US10011607, 50 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  74nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402250BDBM402250(US10011607, 78 | (9aS)-7-[2-chloro-6-fluoro-4-(2- ...)
Affinity DataEC50:  75nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402269BDBM402269(US10011607, 97 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  76nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402226BDBM402226(US10011607, 55 | 2-[(9aRS)-7-[2,6-difluoro-4-(2- p...)
Affinity DataEC50:  77nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402210BDBM402210(US10011607, 41 | (9aS)-2-(2-benzyloxypyrimidin- 5-...)
Affinity DataEC50:  81nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402168BDBM402168(US10011607, 2 | (9aRS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  85nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402238BDBM402238(US10011607, 66 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  85nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402203BDBM402203(US10011607, 36 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  86nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402259BDBM402259(US10011607, 87 | (9aRS)-2-[(2-chloro- phenyl)methy...)
Affinity DataEC50:  87nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402224BDBM402224(US10011607, 53 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  88nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402198BDBM402198(US10011607, 31 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  88nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402199BDBM402199(US10011607, 32 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  88nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402240BDBM402240(US10011607, 68 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  90nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402202BDBM402202(US10011607, 35 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  91nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402237BDBM402237(US10011607, 65 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  92nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402278BDBM402278(US10011607, 106 | (9aS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  95nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402208BDBM402208(US10011607, 39 | (9aS or 9aR)-7-[2,6-difluoro-4-(2...)
Affinity DataEC50:  96nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402243BDBM402243(US10011607, 71 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  101nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402246BDBM402246(US10011607, 74 | (9aRS)-7-[2-chloro-6-fluoro-4-(2-...)
Affinity DataEC50:  102nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402231BDBM402231(US10011607, 59 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  104nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402279BDBM402279(US10011607, 107 | (9aS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  104nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402249BDBM402249(US10011607, 77 | (9aRS)-7-[2-chloro-6-fluoro-4-(2-...)
Affinity DataEC50:  104nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402188BDBM402188(US10011607, 22 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  105nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402180BDBM402180(US10011607, 14 | (9aRS)-7-(2,6-difluoro-4- (phenyl...)
Affinity DataEC50:  105nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402229BDBM402229(US10011607, 57 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  108nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402253BDBM402253(US10011607, 81 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  112nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402209BDBM402209(US10011607, 40 | (9aS)-7-[2,6-difluoro-4-(2- pheny...)
Affinity DataEC50:  113nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402239BDBM402239(US10011607, 67 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  113nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402223BDBM402223(US10011607, 52 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  113nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402197BDBM402197(US10011607, 30 | (9aRS)-7-[2,6-difluoro-4-(2- phen...)
Affinity DataEC50:  113nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 402184BDBM402184(US10011607, 18 | (9aRS)-2-(2-chloro-4-pyridyl)- 7-...)
Affinity DataEC50:  114nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated; for the work with mGlu4 Positive A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details
US Patent

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