Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 898
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297485BDBM297485(US10117944, Compound SDC-TRAP-0249)
Affinity DataIC50: 36nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297487BDBM297487(US10117944, Compound SDC-TRAP-0247)
Affinity DataIC50: 36nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297478BDBM297478(US10117944, Compound SDC-TRAP-0248)
Affinity DataIC50: 37nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297479BDBM297479(US10117944, Compound SDC-TRAP-0244)
Affinity DataIC50: 100nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297482BDBM297482(US10117944, Compound SDC-TRAP-0246)
Affinity DataIC50: 110nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297490BDBM297490(US10117944, Compound SDC-TRAP-0245)
Affinity DataIC50: 117nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297491BDBM297491(US10117944, Compound SDC-TRAP-0242)
Affinity DataIC50: 407nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297481BDBM297481(US10117944, Compound SDC-TRAP-0236)
Affinity DataIC50: 710nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297486BDBM297486(US10117944, Compound SDC-TRAP-0250)
Affinity DataIC50: 2.12E+3nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297489BDBM297489(US10117944, Compound SDC-TRAP-0240)
Affinity DataIC50: 5.00E+3nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297480BDBM297480(US10117944, Compound SDC-TRAP-0237)
Affinity DataIC50: 5.00E+3nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297483BDBM297483(US10117944, Compound SDC-TRAP-0238)
Affinity DataIC50: 5.00E+3nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297484BDBM297484(US10117944, Compound SDC-TRAP-0239)
Affinity DataIC50: 5.00E+3nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Madrigal Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 297488BDBM297488(US10117944, Compound SDC-TRAP-0251)
Affinity DataIC50: 5.00E+3nMAssay Description:HER2 has emerged as a key target for anticancer drugs due to its intrinsic involvement in the phosphatidylinositol-3-kinase-Akt/protein kinase B (PI3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/11/2019
Entry Details
US Patent