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Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 1169
TargetDipeptidyl peptidase 4(Human)
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 311858BDBM311858(US10155775, Example 4 | US10822319, represented by...)
Affinity DataIC50: 2.60nMAssay Description:1. DPP-IV enzyme reaction buffer was prepared (50 mM HEPES (pH=7.8), 80 mM MgCl2, 150 mM NaCl, 1% BSA), and stored on ice for use; 2. The test compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 311861BDBM311861(US10155775, Example 9)
Affinity DataIC50: 3.20nMAssay Description:1. DPP-IV enzyme reaction buffer was prepared (50 mM HEPES (pH=7.8), 80 mM MgCl2, 150 mM NaCl, 1% BSA), and stored on ice for use; 2. The test compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 311860BDBM311860(US10155775, Example 8)
Affinity DataIC50: 3.80nMAssay Description:1. DPP-IV enzyme reaction buffer was prepared (50 mM HEPES (pH=7.8), 80 mM MgCl2, 150 mM NaCl, 1% BSA), and stored on ice for use; 2. The test compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50003020BDBM50003020(MK-3102 | OMARIGLIPTIN | US10155775, Omarigliptin ...)
Affinity DataIC50: 4.20nMAssay Description:1. DPP-IV enzyme reaction buffer was prepared (50 mM HEPES (pH=7.8), 80 mM MgCl2, 150 mM NaCl, 1% BSA), and stored on ice for use; 2. The test compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 311855BDBM311855(US10155775, Example 1)
Affinity DataIC50: 4.40nMAssay Description:1. DPP-IV enzyme reaction buffer was prepared (50 mM HEPES (pH=7.8), 80 mM MgCl2, 150 mM NaCl, 1% BSA), and stored on ice for use; 2. The test compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 311856BDBM311856(US10155775, Example 2)
Affinity DataIC50: 5.10nMAssay Description:1. DPP-IV enzyme reaction buffer was prepared (50 mM HEPES (pH=7.8), 80 mM MgCl2, 150 mM NaCl, 1% BSA), and stored on ice for use; 2. The test compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 311859BDBM311859(US10155775, Example 6)
Affinity DataIC50: 6.5nMAssay Description:1. DPP-IV enzyme reaction buffer was prepared (50 mM HEPES (pH=7.8), 80 mM MgCl2, 150 mM NaCl, 1% BSA), and stored on ice for use; 2. The test compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 311857BDBM311857(US10155775, Example 3)
Affinity DataIC50: 18.2nMAssay Description:1. DPP-IV enzyme reaction buffer was prepared (50 mM HEPES (pH=7.8), 80 mM MgCl2, 150 mM NaCl, 1% BSA), and stored on ice for use; 2. The test compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent