Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 1390
TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320267BDBM320267(US10174023, Compound (5) | 4-(4-fluoro-3-(4-(2-oxo...)
Affinity DataIC50: 1nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320266BDBM320266(US10174023, Compound (4) | 4-(3-(4-(1H-imidazo[4,5...)
Affinity DataIC50: 1nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320275BDBM320275(US10174023, Compound (13) | 4-(3-(4-(1H-imidazo[4,...)
Affinity DataIC50: 1nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320277BDBM320277(US10174023, Compound (15) | 4-(3-(4-(1H-imidazo[4,...)
Affinity DataIC50: 2nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320263BDBM320263(US10174023, Compound (1) | 4-(3-(4-(1H[1,2,3]triaz...)
Affinity DataIC50: 2nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320282BDBM320282(US10174023, Compound (20) | 4-(3-(4-(3H-imidazo[4,...)
Affinity DataIC50: 2nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320271BDBM320271(US10174023, Compound (9) | 4-(3-(4-(2-carbonyl-2,3...)
Affinity DataIC50: 2nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320268BDBM320268(US10174023, Compound (6) | 4-(3-(4-(3H-imidazo[4,5...)
Affinity DataIC50: 3nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320276BDBM320276(US10174023, Compound (14) | 4-(3-(4-(1H-imidazo[4,...)
Affinity DataIC50: 4nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320272BDBM320272(US10174023, Compound (10) | 4-(3-(4-(1H-[1,2,3]tri...)
Affinity DataIC50: 5nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320279BDBM320279(US10174023, Compound (17) | 4-(3-(4-(2-oxo-2,3-dih...)
Affinity DataIC50: 6nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320265BDBM320265(US10174023, Compound (3) | 4-(4-fluoro-3-(4-(2-tri...)
Affinity DataIC50: 6nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320278BDBM320278(US10174023, Compound (16) | 4-(3-(4-(1H-[1,2,3]tri...)
Affinity DataIC50: 7nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320281BDBM320281(US10174023, Compound (19) | 4-(3-(4-(3H-imidazo[4,...)
Affinity DataIC50: 8nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320269BDBM320269(US10174023, Compound (7) | 4-(3-(4-(3H-imidazo[4,5...)
Affinity DataIC50: 8nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 27566BDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)
Affinity DataIC50: 8nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320264BDBM320264(US10174023, Compound (2) | 4-(4-fluoro-3-(4-(2-met...)
Affinity DataIC50: 9nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320274BDBM320274(US10174023, Compound (12) | 4-(3-(4-(2-trifluorome...)
Affinity DataIC50: 10nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320270BDBM320270(US10174023, Compound (8) | 4-(3-(4-(7H-purin-2-yl)...)
Affinity DataIC50: 11nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320280BDBM320280(US10174023, Compound (18) | 4-(3-(4-(3H-imidazo[4,...)
Affinity DataIC50: 13nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320283BDBM320283(US10174023, Compound (21) | 4-(3-(4-(3H-imidazo[4,...)
Affinity DataIC50: 15nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Shanghai Huilun Life Science & Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 320273BDBM320273(US10174023, Compound (11) | 4-(3-(4-(2-methyl-1H-i...)
Affinity DataIC50: 17nMAssay Description:HT Universal Chemiluminescent PARP Assay Kit with Histone-coated Strip Wells, commercially available from Trevigen (US), Catalog #: 4676-096-K.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent