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Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 1920
TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347308BDBM347308(US10202418, Compound A21)
Affinity DataIC50: 24nMAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347290BDBM347290(US10202418, Compound A2)
Affinity DataIC50: 41nMAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347304BDBM347304(US10202418, Compound A17 | US10202418, Compound A1...)
Affinity DataIC50: 255nMAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347289BDBM347289(US10202418, Compound A1)
Affinity DataIC50: 320nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347309BDBM347309(US10202418, Compound A22)
Affinity DataIC50: 350nMAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347289BDBM347289(US10202418, Compound A1)
Affinity DataIC50: 430nMAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347290BDBM347290(US10202418, Compound A2)
Affinity DataIC50: 1.10E+3nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347292BDBM347292(US10202418, Compound A4)
Affinity DataIC50: 4.00E+3nMAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347300BDBM347300(US10202418, Compound A13)
Affinity DataIC50: 4.30E+3nMAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetCathepsin D(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347294BDBM347294(US10202418, Compound A6)
Affinity DataIC50: 1.20E+4nMAssay Description:In order to identify modulators of cathepsin D activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluores...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347308BDBM347308(US10202418, Compound A21)
Affinity DataIC50: 1.20E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347291BDBM347291(US10202418, Compound A3)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347293BDBM347293(US10202418, Compound A5)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347292BDBM347292(US10202418, Compound A4)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347309BDBM347309(US10202418, Compound A22)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347303BDBM347303(US10202418, Compound A16)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347301BDBM347301(US10202418, Compound A14)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347302BDBM347302(US10202418, Compound A15)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347306BDBM347306(US10202418, Compound A19)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347307BDBM347307(US10202418, Compound A20)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347304BDBM347304(US10202418, Compound A17 | US10202418, Compound A1...)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347304BDBM347304(US10202418, Compound A17 | US10202418, Compound A1...)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347296BDBM347296(US10202418, Compound A8)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347297BDBM347297(US10202418, Compound A9)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347294BDBM347294(US10202418, Compound A6)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347295BDBM347295(US10202418, Compound A7)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347300BDBM347300(US10202418, Compound A13)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347298BDBM347298(US10202418, Compound A10)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent

TargetRenin(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 347299BDBM347299(US10202418, Compound A12)
Affinity DataIC50: 3.00E+4nMAssay Description:In order to identify modulators of renin activity, a continuous enzymatic test was carried out with a synthetic peptide which carries a fluorescent g...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2019
Entry Details
US Patent