Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 2321
TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361601BDBM361601(US10221175, Compound 6)
Affinity DataEC50:  488nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361604BDBM361604(A. Preparation of 7-(2-fluoro-4-(2-methyl-2H-indaz...)
Affinity DataEC50:  502nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361612BDBM361612(US10221175, Compound 17)
Affinity DataEC50:  618nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361598BDBM361598(US10221175, Compound 3)
Affinity DataEC50:  656nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361625BDBM361625(US10221175, Compound 30)
Affinity DataEC50:  677nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361597BDBM361597(A. Preparation of 7-(2-fluoro-4-(2-methyl-2H-indaz...)
Affinity DataEC50:  688nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361600BDBM361600(US10221175, Compound 5)
Affinity DataEC50:  743nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361606BDBM361606(US10221175, Compound 11)
Affinity DataEC50:  856nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361634BDBM361634(US10221175, Compound 39)
Affinity DataEC50:  857nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361596BDBM361596(A. Preparation of 7-(2,6-difluoro-4-(2-methyl-2h-i...)
Affinity DataEC50:  952nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361603BDBM361603(US10221175, Compound 8)
Affinity DataEC50:  1.06E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361611BDBM361611(US10221175, Compound 16)
Affinity DataEC50:  1.21E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361610BDBM361610(US10221175, Compound 15)
Affinity DataEC50:  1.24E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361617BDBM361617(US10221175, Compound 22)
Affinity DataEC50:  1.31E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361618BDBM361618(US10221175, Compound 23)
Affinity DataEC50:  1.35E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361627BDBM361627(US10221175, Compound 32)
Affinity DataEC50:  1.40E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361614BDBM361614(US10221175, Compound 19)
Affinity DataEC50:  1.41E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361605BDBM361605(US10221175, Compound 10)
Affinity DataEC50:  1.57E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361626BDBM361626(US10221175, Compound 31)
Affinity DataEC50:  1.63E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361599BDBM361599(US10221175, Compound 4)
Affinity DataEC50:  1.75E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361609BDBM361609(US10221175, Compound 14)
Affinity DataEC50:  1.79E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361608BDBM361608(US10221175, Compound 13)
Affinity DataEC50:  1.82E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361615BDBM361615(US10221175, Compound 20)
Affinity DataEC50:  2.10E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361613BDBM361613(US10221175, Compound 18)
Affinity DataEC50:  2.14E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361628BDBM361628(US10221175, Compound 33)
Affinity DataEC50:  2.20E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361622BDBM361622(US10221175, Compound 27)
Affinity DataEC50:  2.26E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361623BDBM361623(US10221175, Compound 28)
Affinity DataEC50:  2.37E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361602BDBM361602(US10221175, Compound 7)
Affinity DataEC50:  2.64E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361629BDBM361629(US10221175, Compound 34)
Affinity DataEC50:  3.90E+3nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361630BDBM361630(US10221175, Compound 35)
Affinity DataEC50:  1.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361631BDBM361631(US10221175, Compound 36)
Affinity DataEC50:  1.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361635BDBM361635(US10221175, Compound 40)
Affinity DataEC50:  1.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361616BDBM361616(US10221175, Compound 21)
Affinity DataEC50:  1.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361632BDBM361632(US10221175, Compound 37)
Affinity DataEC50:  1.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361633BDBM361633(US10221175, Compound 38)
Affinity DataEC50:  1.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361636BDBM361636(US10221175, Compound 41)
Affinity DataEC50:  1.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361637BDBM361637(US10221175, Compound 42)
Affinity DataEC50:  1.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361624BDBM361624(US10221175, Compound 29)
Affinity DataEC50:  3.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361619BDBM361619(US10221175, Compound 24)
Affinity DataEC50:  3.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361607BDBM361607(US10221175, Compound 12)
Affinity DataEC50:  3.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361620BDBM361620(US10221175, Compound 25)
Affinity DataEC50:  3.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 361621BDBM361621(US10221175, Compound 26)
Affinity DataEC50:  3.00E+4nMAssay Description:For high throughput measurement of agonist-evoked increases in intracellular calcium, CHO-K1 cells stably expressing muscarinic receptors were plated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2019
Entry Details
US Patent