Compile Data Set for Download or QSAR
Report error Found 116 Enz. Inhib. hit(s) with all data for entry = 2751
TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086441BDBM50086441(CHEMBL3426225 | US10266537, Compound 3)
Affinity DataIC50: 1nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Yes(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 1nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Yes(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378887BDBM378887(US10266537, Compound 31)
Affinity DataIC50: 1nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Yes(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086441BDBM50086441(CHEMBL3426225 | US10266537, Compound 3)
Affinity DataIC50: 1nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Yes(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378888BDBM378888(US10266537, Compound 120 | Preparation of 3-(4-ami...)
Affinity DataIC50: 1nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086441BDBM50086441(CHEMBL3426225 | US10266537, Compound 3)
Affinity DataIC50: 1nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetBreakpoint cluster region protein [1-693](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086441BDBM50086441(CHEMBL3426225 | US10266537, Compound 3)
Affinity DataIC50: 1nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 2nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Yes(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086442BDBM50086442(CHEMBL3426233 | US10266537, Compound 121)
Affinity DataIC50: 2nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378887BDBM378887(US10266537, Compound 31)
Affinity DataIC50: 2nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378890BDBM378890(US10266537, Compound 5)
Affinity DataIC50: 2nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase ABL1 [T315I](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 3nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase HCK(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 3nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086441BDBM50086441(CHEMBL3426225 | US10266537, Compound 3)
Affinity DataIC50: 3nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Fyn(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378887BDBM378887(US10266537, Compound 31)
Affinity DataIC50: 3nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086453BDBM50086453(CHEMBL3426220 | US10266537, Compound 14)
Affinity DataIC50: 3nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 3nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Lyn(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 4nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetHepatocyte growth factor receptor(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 4nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086456BDBM50086456(CHEMBL3426218 | US10266537, Compound 17)
Affinity DataIC50: 4nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378889BDBM378889(US10266537, Compound 1 | Preparation of N-(3-((4-a...)
Affinity DataIC50: 4nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase ABL2(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 4nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378902BDBM378902(US10266537, Compound 18)
Affinity DataIC50: 4nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378887BDBM378887(US10266537, Compound 31)
Affinity DataIC50: 4nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Fyn(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086441BDBM50086441(CHEMBL3426225 | US10266537, Compound 3)
Affinity DataIC50: 5nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetSerine/threonine-protein kinase B-raf [V600E](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378887BDBM378887(US10266537, Compound 31)
Affinity DataIC50: 5nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086586BDBM50086586(CHEMBL3426234 | US10266537, Compound 29)
Affinity DataIC50: 5nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Fyn(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 6nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetCytoplasmic tyrosine-protein kinase BMX(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086441BDBM50086441(CHEMBL3426225 | US10266537, Compound 3)
Affinity DataIC50: 6nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 7nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378900BDBM378900(US10266537, Compound 16)
Affinity DataIC50: 7nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086445BDBM50086445(CHEMBL3426229 | US10266537, Compound 21)
Affinity DataIC50: 7nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086444BDBM50086444(CHEMBL3426230 | US10266537, Compound 20)
Affinity DataIC50: 7nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086449BDBM50086449(CHEMBL3426224 | US10266537, Compound 8)
Affinity DataIC50: 7nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetSerine/threonine-protein phosphatase(Yeast)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 8nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086446BDBM50086446(CHEMBL3426228 | US10266537, Compound 19)
Affinity DataIC50: 8nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetEpidermal growth factor receptor [T790M,L858R](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 8nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase CSK(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 9nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086441BDBM50086441(CHEMBL3426225 | US10266537, Compound 3)
Affinity DataIC50: 9nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086448BDBM50086448(CHEMBL3426226 | US10266537, Compound 6)
Affinity DataIC50: 9nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378896BDBM378896(US10266537, Compound 11)
Affinity DataIC50: 10nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetEphrin type-B receptor 2(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378887BDBM378887(US10266537, Compound 31)
Affinity DataIC50: 10nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetAngiopoietin-1 receptor(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378885BDBM378885(US10266537, Compound 93)
Affinity DataIC50: 10nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378898BDBM378898(US10266537, Compound 13)
Affinity DataIC50: 11nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetEphrin type-B receptor 4(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378887BDBM378887(US10266537, Compound 31)
Affinity DataIC50: 11nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetCytoplasmic tyrosine-protein kinase BMX(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378888BDBM378888(US10266537, Compound 120 | Preparation of 3-(4-ami...)
Affinity DataIC50: 11nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 50086585BDBM50086585(CHEMBL3426235 | US10266537, Compound 26)
Affinity DataIC50: 11nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src [1-530](Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378888BDBM378888(US10266537, Compound 120 | Preparation of 3-(4-ami...)
Affinity DataIC50: 12nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetTyrosine-protein kinase Blk(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378887BDBM378887(US10266537, Compound 31)
Affinity DataIC50: 12nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
St. Chuan University

US Patent
LigandChemical structure of BindingDB Monomer ID 378887BDBM378887(US10266537, Compound 31)
Affinity DataIC50: 12nMAssay Description:The aim of this experiment is to detect the inhibitory activity of the compounds of the present invention against in vitro protein kinases using isot...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2020
Entry Details
US Patent

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