Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 3527
TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403299BDBM403299(US10329307, Example 46)
Affinity DataIC50: 240nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403270BDBM403270(US10329307, Example 17)
Affinity DataIC50: 290nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403298BDBM403298(US10329307, Example 45)
Affinity DataIC50: 370nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403263BDBM403263(US10329307, Example 10)
Affinity DataIC50: 390nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403254BDBM403254(US10329307, Example 1)
Affinity DataIC50: 420nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403265BDBM403265(US10329307, Example 12)
Affinity DataIC50: 420nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403286BDBM403286(US10329307, Example 33)
Affinity DataIC50: 440nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403275BDBM403275(US10329307, Example 22)
Affinity DataIC50: 440nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403272BDBM403272(US10329307, Example 19)
Affinity DataIC50: 460nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403271BDBM403271(US10329307, Example 18)
Affinity DataIC50: 470nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403296BDBM403296(US10329307, Example 43)
Affinity DataIC50: 480nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403269BDBM403269(US10329307, Example 16)
Affinity DataIC50: 500nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403292BDBM403292(US10329307, Example 39)
Affinity DataIC50: 510nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403274BDBM403274(US10329307, Example 21)
Affinity DataIC50: 540nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403291BDBM403291(US10329307, Example 38)
Affinity DataIC50: 540nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403266BDBM403266(US10329307, Example 13)
Affinity DataIC50: 550nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403290BDBM403290(US10329307, Example 37)
Affinity DataIC50: 560nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403276BDBM403276(US10329307, Example 23)
Affinity DataIC50: 600nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403287BDBM403287(US10329307, Example 34)
Affinity DataIC50: 700nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403273BDBM403273(US10329307, Example 20)
Affinity DataIC50: 710nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403308BDBM403308(US10329307, Example 55 | US10329307, Example 57 | ...)
Affinity DataIC50: 720nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403264BDBM403264(US10329307, Example 11)
Affinity DataIC50: 740nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403308BDBM403308(US10329307, Example 55 | US10329307, Example 57 | ...)
Affinity DataIC50: 740nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403297BDBM403297(US10329307, Example 44)
Affinity DataIC50: 750nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403289BDBM403289(US10329307, Example 36)
Affinity DataIC50: 750nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403278BDBM403278(US10329307, Example 25)
Affinity DataIC50: 790nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403316BDBM403316(US10329307, Example 63 | US10329307, Example 65 | ...)
Affinity DataIC50: 820nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403288BDBM403288(US10329307, Example 35)
Affinity DataIC50: 840nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403316BDBM403316(US10329307, Example 63 | US10329307, Example 65 | ...)
Affinity DataIC50: 860nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403283BDBM403283(US10329307, Example 30)
Affinity DataIC50: 860nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403284BDBM403284(US10329307, Example 31)
Affinity DataIC50: 890nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403308BDBM403308(US10329307, Example 55 | US10329307, Example 57 | ...)
Affinity DataIC50: 920nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403282BDBM403282(US10329307, Example 29)
Affinity DataIC50: 950nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403277BDBM403277(US10329307, Example 24)
Affinity DataIC50: 950nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403262BDBM403262(US10329307, Example 9)
Affinity DataIC50: 950nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403300BDBM403300(US10329307, Example 47)
Affinity DataIC50: 1.00E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403316BDBM403316(US10329307, Example 63 | US10329307, Example 65 | ...)
Affinity DataIC50: 1.00E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403301BDBM403301(US10329307, Example 48)
Affinity DataIC50: 1.10E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403295BDBM403295(US10329307, Example 42)
Affinity DataIC50: 1.10E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403305BDBM403305(US10329307, Example 52)
Affinity DataIC50: 1.10E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403312BDBM403312(US10329307, Example 59)
Affinity DataIC50: 1.20E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403256BDBM403256(US10329307, Example 3)
Affinity DataIC50: 1.20E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403268BDBM403268(US10329307, Example 15)
Affinity DataIC50: 1.30E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403324BDBM403324(US10329307, Example 71)
Affinity DataIC50: 1.30E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403293BDBM403293(US10329307, Example 40)
Affinity DataIC50: 1.30E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403319BDBM403319(US10329307, Example 66)
Affinity DataIC50: 1.40E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403325BDBM403325(US10329307, Example 72)
Affinity DataIC50: 1.40E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403261BDBM403261(US10329307, Example 8)
Affinity DataIC50: 1.40E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403279BDBM403279(US10329307, Example 26)
Affinity DataIC50: 1.40E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

TargetPRKC apoptosis WT1 regulator protein(Human)
Universite De Montreal

US Patent
LigandChemical structure of BindingDB Monomer ID 403311BDBM403311(US10329307, Example 58)
Affinity DataIC50: 1.40E+3nMAssay Description:FLIPR-based calcium mobilization assay in HEK293 cells was used to measure PAR4 antagonism, agonism, and selectivity against PAR1. The activity of th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/31/2020
Entry Details
US Patent

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