Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 8773
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Algiax Pharmaceuticals

US Patent
LigandPNGBDBM419906(US10472324, Example 9)
Affinity DataIC50: 5.00E+3nMAssay Description:The affinity of the test compounds for the GABA gated Cl-channel (GABA.A receptor complex) in the rat cerebral cortex was determined in a radioligand...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/14/2020
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Algiax Pharmaceuticals

US Patent
LigandPNGBDBM419122(US10472324, Example 1)
Affinity DataIC50: 5.30E+3nMAssay Description:The affinity of the test compounds for the GABA gated Cl-channel (GABA.A receptor complex) in the rat cerebral cortex was determined in a radioligand...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2020
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Algiax Pharmaceuticals

US Patent
LigandPNGBDBM419852(US10472324, Example 3)
Affinity DataIC50: 6.00E+3nMAssay Description:The affinity of the test compounds for the GABA gated Cl-channel (GABA.A receptor complex) in the rat cerebral cortex was determined in a radioligand...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/14/2020
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Algiax Pharmaceuticals

US Patent
LigandPNGBDBM419902(US10472324, Example 5)
Affinity DataIC50: 7.70E+3nMAssay Description:The affinity of the test compounds for the GABA gated Cl-channel (GABA.A receptor complex) in the rat cerebral cortex was determined in a radioligand...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/14/2020
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Algiax Pharmaceuticals

US Patent
LigandPNGBDBM419903(US10472324, Example 6)
Affinity DataIC50: 7.90E+3nMAssay Description:The affinity of the test compounds for the GABA gated Cl-channel (GABA.A receptor complex) in the rat cerebral cortex was determined in a radioligand...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/14/2020
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Algiax Pharmaceuticals

US Patent
LigandPNGBDBM419125(US10472324, Example 2)
Affinity DataIC50: 8.30E+3nMAssay Description:The affinity of the test compounds for the GABA gated Cl-channel (GABA.A receptor complex) in the rat cerebral cortex was determined in a radioligand...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/14/2020
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Algiax Pharmaceuticals

US Patent
LigandPNGBDBM419901(US10472324, Example 4)
Affinity DataIC50: 8.70E+3nMAssay Description:The affinity of the test compounds for the GABA gated Cl-channel (GABA.A receptor complex) in the rat cerebral cortex was determined in a radioligand...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/14/2020
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Algiax Pharmaceuticals

US Patent
LigandPNGBDBM419904(US10472324, Example 7)
Affinity DataIC50: 9.60E+3nMAssay Description:The affinity of the test compounds for the GABA gated Cl-channel (GABA.A receptor complex) in the rat cerebral cortex was determined in a radioligand...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/14/2020
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Algiax Pharmaceuticals

US Patent
LigandPNGBDBM419905(US10472324, Example 8)
Affinity DataIC50: 1.03E+4nMAssay Description:The affinity of the test compounds for the GABA gated Cl-channel (GABA.A receptor complex) in the rat cerebral cortex was determined in a radioligand...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/14/2020
Entry Details
US Patent