Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 8821
TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420962(US10479798, Compound 21)
Affinity DataIC50: 2nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoPDBSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM50198186(CHEMBL3944427 | US10479798, Compound 19)
Affinity DataIC50: 2nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM50003020(MK-3102 | OMARIGLIPTIN | US10155775, Omarigliptin ...)
Affinity DataIC50: 2nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420415(US10479798, Compound 12)
Affinity DataIC50: 4nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM50198175(CHEMBL3932825 | US10479798, Compound 17)
Affinity DataIC50: 6nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420402(US10479798, Compound 9)
Affinity DataIC50: 9.17nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420956(US10479798, Compound 16)
Affinity DataIC50: 11nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 14nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM50198180(CHEMBL3928073 | US10479798, Compound 5)
Affinity DataIC50: 15nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420408(US10479798, Compound 10)
Affinity DataIC50: 18nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM50198178(CHEMBL3901191 | US10479798, Compound 6)
Affinity DataIC50: 20nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM50198184(CHEMBL3942843 | US10479798, Compound 20)
Affinity DataIC50: 30nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420966(US10479798, Compound 25)
Affinity DataIC50: 33nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM50198185(CHEMBL3979508 | US10479798, Compound 7)
Affinity DataIC50: 39nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420971(US10479798, Compound 30)
Affinity DataIC50: 55nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420969(US10479798, Compound 28)
Affinity DataIC50: 56nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420958(US10479798, Compound 18)
Affinity DataIC50: 70nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420477(US10479798, Compound 14)
Affinity DataIC50: 74nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420965(US10479798, Compound 24)
Affinity DataIC50: 78nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420854(US10479798, Compound 15)
Affinity DataIC50: 110nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM50198164(CHEMBL3959577 | US10479798, Compound 3)
Affinity DataIC50: 154nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420453(US10479798, Compound 13)
Affinity DataIC50: 169nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420412(US10479798, Compound 11)
Affinity DataIC50: 205nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420328(US10479798, Compound 2)
Affinity DataIC50: 207nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420400(US10479798, Compound 8)
Affinity DataIC50: 216nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420970(US10479798, Compound 29)
Affinity DataIC50: 254nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420338(US10479798, Compound 4)
Affinity DataIC50: 283nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420967(US10479798, Compound 26)
Affinity DataIC50: 338nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420963(US10479798, Compound 22)
Affinity DataIC50: 564nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420968(US10479798, Compound 27)
Affinity DataIC50: 678nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420964(US10479798, Compound 23)
Affinity DataIC50: 800nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandPNGBDBM420322(US10479798, Compound 1)
Affinity DataIC50: 3.32E+3nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent