Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 8954
TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431919BDBM431919(((S)-6-{(R)-4-[2,6-Dimethyl-4-(2-methyl-2H-tetrazo...)
Affinity DataEC50:  6nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431921BDBM431921(((S)-6-{(R)-4-[2,6-Dimethyl-4-(2-methyl-2H-tetrazo...)
Affinity DataEC50:  7nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431934BDBM431934({(S)-6-[(R)-4-(2,6-Dimethyl-4-pyrazin-2-yl-phenyl)...)
Affinity DataEC50:  9nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431929BDBM431929([(S)-6-((R)-7-Fluoro-4-{4-[2-(2-hydroxo-2-methyl-p...)
Affinity DataEC50:  9nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431931BDBM431931(((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-2-oxo-1,2-...)
Affinity DataEC50:  12nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431932BDBM431932(((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-6-oxo-1,6-...)
Affinity DataEC50:  14nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431915BDBM431915(((S)-6-{(R)-7-Fluoro-4-[4-(3-hydroxy-3-methyl-buto...)
Affinity DataEC50:  15nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431917BDBM431917(((S)-6-{(R)-4-[4-(3-Hydroxy-3-methyl-butoxy)-2,6-d...)
Affinity DataEC50:  21nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431933BDBM431933(((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-6-oxo-1,6-...)
Affinity DataEC50:  27nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431930BDBM431930(((S)-6-{(R)-4-[2,6-Dimethyl-4-(1-methyl-2-oxo-1,2-...)
Affinity DataEC50:  27nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431928BDBM431928(((S)-6-{(R)-4-[2,6-Dimethyl-4-(tetrahydro-furan-3-...)
Affinity DataEC50:  27nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431927BDBM431927(((S)-6-{(R)-7-Fluoro-4-[4-(2-hydroxo-2-methyl-prop...)
Affinity DataEC50:  35nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431925BDBM431925(((S)-6-{(R)-4-[2,6-Dimethyl-4-(3-methyl-oxetan-3-y...)
Affinity DataEC50:  37nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431924BDBM431924(((S)-6-{(R)-4-[2,6-Dimethyl-4-(tetrahydro-pyran-4-...)
Affinity DataEC50:  56nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431923BDBM431923([(S)-6-((R)-4-{2,6-Dimethyl-4-[(R)-(tetrahydro-fur...)
Affinity DataEC50:  57nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431926BDBM431926([(S)-6-((R)-4-{2,6-Dimethyl-4-[(S)-(tetrahydro-fur...)
Affinity DataEC50:  73nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431922BDBM431922(((R)-6-{(R)-4-[2,6-Dimethyl-4-(2-methyl-2H-tetrazo...)
Affinity DataEC50:  378nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431920BDBM431920(((R)-6-{(R)-4-[2,6-Dimethyl-4-(2-methyl-2H-tetrazo...)
Affinity DataEC50:  382nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431918BDBM431918(((R)-6-{(R)-4-[4-(3-Hydroxy-3-methyl-butoxy)-2,6-d...)
Affinity DataEC50:  751nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetFree fatty acid receptor 1(Human)
Boehringer Ingelheim International

US Patent
LigandChemical structure of BindingDB Monomer ID 431916BDBM431916(((R)-6-{(R)-7-Fluoro-4-[4-(3-hydroxy-3-methyl-buto...)
Affinity DataEC50:  764nMAssay Description:IP1 accumulation measurements using the IPOne assay system 1321N1 cells stably expressing human GPR40 receptor (Euroscreen, Belgium) are seeded 24 h ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent