Compile Data Set for Download or QSAR
Report error Found 112 Enz. Inhib. hit(s) with all data for entry = 9072
TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439120(US10604502, Ex # 108)
Affinity DataIC50: 1nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439100(US10604502, Ex # 88)
Affinity DataIC50: 1nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439039(US10604502, Ex # 27)
Affinity DataIC50: 2nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439089(US10604502, Ex # 77)
Affinity DataIC50: 2nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439014(US10604502, Ex # 2)
Affinity DataIC50: 2nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439109(3-(2,2-dimethyl-1,2,3,4-tetrahydroquinolin-5-yl)-1...)
Affinity DataIC50: 3nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439056(US10604502, Ex # 44)
Affinity DataIC50: 4nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439101(3-(2,2-dimethyl-1,2,3,4-tetrahydro-1,7-naphthyridi...)
Affinity DataIC50: 4nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439046(US10604502, Ex # 34)
Affinity DataIC50: 4nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439090(US10604502, Ex # 78)
Affinity DataIC50: 5nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439121(1-((1R,4R)-1-aminosulfonylcyclohexyl)-6-methyl-3-(...)
Affinity DataIC50: 5nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439036(3-(3-amino-2-methylphenyl)-1-(3-hydroxypropyl)-2,6...)
Affinity DataIC50: 5nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439015(US10604502, Ex # 3)
Affinity DataIC50: 5nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439107(US10604502, Ex # 95)
Affinity DataIC50: 5nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439024(US10604502, Ex # 12)
Affinity DataIC50: 6nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439122(US10604502, Ex # 110)
Affinity DataIC50: 6nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439021(US10604502, Ex # 9)
Affinity DataIC50: 6nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439059(US10604502, Ex # 47)
Affinity DataIC50: 6nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439091(US10604502, Ex # 79)
Affinity DataIC50: 6nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439124(1-((1R,4R)-4-cyanocyclohexyl)-6-methyl-3-(5-amino-...)
Affinity DataIC50: 8nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439123(US10604502, Ex # 111)
Affinity DataIC50: 8nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439079(US10604502, Ex # 67)
Affinity DataIC50: 9nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439108(US10604502, Ex # 96)
Affinity DataIC50: 9nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439092(3-(5-amino-4-chloropyridin-3-yl)-6-methyl-1-(5-(me...)
Affinity DataIC50: 10nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439013(US10604502, Ex # 1)
Affinity DataIC50: 10nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439041(US10604502, Ex # 29)
Affinity DataIC50: 12nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439033(US10604502, Ex # 21)
Affinity DataIC50: 12nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439093(US10604502, Ex # 81)
Affinity DataIC50: 12nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439077(US10604502, Ex # 65)
Affinity DataIC50: 13nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439038(US10604502, Ex # 26)
Affinity DataIC50: 14nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439062(US10604502, Ex # 50)
Affinity DataIC50: 14nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439094(US10604502, Ex # 82)
Affinity DataIC50: 15nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439074(US10604502, Ex # 62)
Affinity DataIC50: 16nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439080(3(3-(5-amino-4-chloropyridin-3-yl)-5-cyano-6-methy...)
Affinity DataIC50: 16nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439044(US10604502, Ex # 32)
Affinity DataIC50: 16nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439022(US10604502, Ex # 10)
Affinity DataIC50: 17nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439069(US10604502, Ex # 57)
Affinity DataIC50: 18nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439064(US10604502, Ex # 52)
Affinity DataIC50: 18nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439086(US10604502, Ex # 74)
Affinity DataIC50: 20nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439066(US10604502, Ex # 54)
Affinity DataIC50: 23nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439075(US10604502, Ex # 63)
Affinity DataIC50: 23nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439026(US10604502, Ex # 14)
Affinity DataIC50: 24nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439047(US10604502, Ex # 35)
Affinity DataIC50: 25nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439110(US10604502, Ex # 98)
Affinity DataIC50: 25nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439057((1R,4R)-4-(3-(5-amino-4-chloropyridin-3-yl)-5-cyan...)
Affinity DataIC50: 26nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439016(US10604502, Ex # 15 | US10604502, Ex # 4)
Affinity DataIC50: 26nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439016(US10604502, Ex # 15 | US10604502, Ex # 4)
Affinity DataIC50: 27nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439023(US10604502, Ex # 11)
Affinity DataIC50: 28nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439019(US10604502, Ex # 7)
Affinity DataIC50: 28nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Novartis

US Patent
LigandPNGBDBM439095(US10604502, Ex # 83)
Affinity DataIC50: 28nMAssay Description:Representative compounds of the present invention were serially and separately diluted 3-fold in DMSO to obtain a total of twelve concentrations. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2020
Entry Details
US Patent

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