Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 9334
LigandChemical structure of BindingDB Monomer ID 458500BDBM458500(2-(2-Fluoro-6-methoxyphenyl)-N-(4-((2-hydroxy-2-me...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458501BDBM458501(2-(2-Fluoro-6-methoxyphenyl)-N-(1-methyl-4-(methyl...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458498BDBM458498(2-(2-Fluoro-6-methoxyphenyl)-N-(1-methyl-4-(methyl...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458499BDBM458499(2-(2-Fluoro-6-methoxyphenyl)-N-(1-methyl-4-(methyl...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458495BDBM458495(N-(4-(Dimethylamino)-1-methyl-1H-indazol-5-yl)-2-(...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458496BDBM458496(N-(4-(Benzyl(methyl)amino)-1-methyl-1H-indazol-5-y...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458490BDBM458490(2-(2-Fluoro-6-methoxyphenyl)-N-(1-methyl-4-(methyl...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458491BDBM458491(N-(4-(Cyclopropyl(methyl)amino)-1-methyl-1H-indazo...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458487BDBM458487(US10745388, Example 1, Peak 1)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458489BDBM458489(US10745388, Example 1, Peak 2)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458506BDBM458506((S) N-(4-((1-(Dimethylcarbamoyl)pyrrolidin-3-yl)(m...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458507BDBM458507(2-(2-Fluoro-6-methoxyphenyl)-N-(1-methyl-4-(2-((me...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458504BDBM458504((S) N-(4-((1-acetylpyrrolidin-3-yl)(methyl)amino)-...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458505BDBM458505((S)-2-(2-Fluoro-6-methoxyphenyl)-N-(1-methyl-4-(me...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458503BDBM458503((S)-2-(2-Fluoro-6-methoxyphenyl)-N-(1-methyl-4-(me...)
Affinity DataKi: <100nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458502BDBM458502(2-(2-Fluoro-6-methoxyphenyl)-N-(4-(((3-hydroxyoxet...)
Affinity DataKi:  2.75E+3nMAssay Description:A stock solution of 1 mM test compound was prepared in DMSO. The compound plate was prepared by 3-fold and 11-point serial dilutions. 0.1 μL of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent