Compile Data Set for Download or QSAR
Report error Found 205 Enz. Inhib. hit(s) with all data for entry = 9534
TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242764BDBM242764(US9422299, 30 | US10030025, Compound 30 | US998727...)
Affinity DataIC50: 5nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242764BDBM242764(US9422299, 30 | US10030025, Compound 30 | US998727...)
Affinity DataKi:  7nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 50112180BDBM50112180(CHEMBL3608688 | US9422299, 41 | US10030025, Compou...)
Affinity DataIC50: 7nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242740BDBM242740(US9422299, 1 | US10030025, Compound 1 | US9987274,...)
Affinity DataKi:  11nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 50112180BDBM50112180(CHEMBL3608688 | US9422299, 41 | US10030025, Compou...)
Affinity DataKi:  11nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242741BDBM242741(US9422299, 2 | US10030025, Compound 2 | US9987274,...)
Affinity DataIC50: 12nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242741BDBM242741(US9422299, 2 | US10030025, Compound 2 | US9987274,...)
Affinity DataKi:  15nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242740BDBM242740(US9422299, 1 | US10030025, Compound 1 | US9987274,...)
Affinity DataIC50: 16nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 50112244BDBM50112244(CHEMBL3608680 | US9422299, 5 | US10030025, Compoun...)
Affinity DataIC50: 18nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 50112181BDBM50112181(CHEMBL3608687 | US9422299, 3 | US10030025, Compoun...)
Affinity DataKi:  19nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242742BDBM242742(US9422299, 4 | US10030025, Compound 4 | US9987274,...)
Affinity DataIC50: 19nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242742BDBM242742(US9422299, 4 | US10030025, Compound 4 | US9987274,...)
Affinity DataKi:  20nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242746BDBM242746(US9422299, 9 | US10030025, Compound 9 | US9987274,...)
Affinity DataIC50: 21nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 50112244BDBM50112244(CHEMBL3608680 | US9422299, 5 | US10030025, Compoun...)
Affinity DataKi:  23nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242743BDBM242743(US9422299, 6 | US10030025, Compound 6 | US9987274,...)
Affinity DataKi:  24nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242772BDBM242772(US9422299, 38 | US10030025, Compound 38 | US998727...)
Affinity DataKi:  26nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242745BDBM242745(US9422299, 8 | US10030025, Compound 8 | US9987274,...)
Affinity DataKi:  26nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242744BDBM242744(US9422299, 7 | US10030025, Compound 7 | US9987274,...)
Affinity DataKi:  26nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242773BDBM242773(US9422299, 39 | US10030025, Compound 39 | US998727...)
Affinity DataKi:  28nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242744BDBM242744(US9422299, 7 | US10030025, Compound 7 | US9987274,...)
Affinity DataIC50: 30nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242743BDBM242743(US9422299, 6 | US10030025, Compound 6 | US9987274,...)
Affinity DataIC50: 30nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242746BDBM242746(US9422299, 9 | US10030025, Compound 9 | US9987274,...)
Affinity DataKi:  30nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242747BDBM242747(US9422299, 10 | US10030025, Compound 10 | US998727...)
Affinity DataKi:  31nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242773BDBM242773(US9422299, 39 | US10030025, Compound 39 | US998727...)
Affinity DataIC50: 32nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 50112245BDBM50112245(CHEMBL3608741 | US9422299, 11 | US10030025, Compou...)
Affinity DataKi:  32nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 50112181BDBM50112181(CHEMBL3608687 | US9422299, 3 | US10030025, Compoun...)
Affinity DataIC50: 32nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242745BDBM242745(US9422299, 8 | US10030025, Compound 8 | US9987274,...)
Affinity DataIC50: 33nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242772BDBM242772(US9422299, 38 | US10030025, Compound 38 | US998727...)
Affinity DataIC50: 34nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242768BDBM242768(US9422299, 34 | US10030025, Compound 34 | US998727...)
Affinity DataKi:  38nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242775BDBM242775(US9422299, 42 | US10030025, Compound 42 | US998727...)
Affinity DataIC50: 39nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242749BDBM242749(US9422299, 13 | US10030025, Compound 13 | US998727...)
Affinity DataKi:  40nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242771BDBM242771(US9422299, 37 | US10030025, Compound 37 | US998727...)
Affinity DataKi:  41nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242750BDBM242750(US9422299, 14 | US10030025, Compound 14 | US998727...)
Affinity DataKi:  42nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242770BDBM242770(US9422299, 36 | US10030025, Compound 36 | US998727...)
Affinity DataKi:  43nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242749BDBM242749(US9422299, 13 | US10030025, Compound 13 | US998727...)
Affinity DataIC50: 44nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242766BDBM242766(US9422299, 32 | US10030025, Compound 32 | US998727...)
Affinity DataIC50: 44nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242777BDBM242777(US9422299, 44 | US10030025, Compound 44 | US998727...)
Affinity DataKi:  45nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242751BDBM242751(US9422299, 15 | US10030025, Compound 15 | US998727...)
Affinity DataKi:  45nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242775BDBM242775(US9422299, 42 | US10030025, Compound 42 | US998727...)
Affinity DataKi:  48nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242752BDBM242752(US9422299, 16 | US10030025, Compound 16 | US998727...)
Affinity DataKi:  49nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242751BDBM242751(US9422299, 15 | US10030025, Compound 15 | US998727...)
Affinity DataIC50: 50nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242753BDBM242753(US9422299, 17 | US10030025, Compound 17 | US998727...)
Affinity DataIC50: 50nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242753BDBM242753(US9422299, 17 | US10030025, Compound 17 | US998727...)
Affinity DataKi:  51nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242771BDBM242771(US9422299, 37 | US10030025, Compound 37 | US998727...)
Affinity DataIC50: 52nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242754BDBM242754(US9422299, 18 | US10030025, Compound 18 | US998727...)
Affinity DataKi:  54nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242769BDBM242769(US9422299, 35 | US10030025, Compound 35 | US998727...)
Affinity DataIC50: 54nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242755BDBM242755(US9422299, 19 | US10030025, Compound 19 | US998727...)
Affinity DataKi:  56nMAssay Description:The affinity of compounds of the invention for the human NK-3 receptor was determined by measuring the ability of compounds of the invention to compe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242747BDBM242747(US9422299, 10 | US10030025, Compound 10 | US998727...)
Affinity DataIC50: 56nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242750BDBM242750(US9422299, 14 | US10030025, Compound 14 | US998727...)
Affinity DataIC50: 57nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

TargetNeuromedin-K receptor(Human)
Ogeda

US Patent
LigandChemical structure of BindingDB Monomer ID 242770BDBM242770(US9422299, 36 | US10030025, Compound 36 | US998727...)
Affinity DataIC50: 58nMAssay Description:Changes in intracellular calcium levels are a recognized indicator of G protein-coupled receptor activity. The efficacy of compounds of the invention...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

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