Compile Data Set for Download or QSAR
Report error Found 103 Enz. Inhib. hit(s) with all data for entry = 9659
TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479434BDBM479434(US10894807, ID P242)
Affinity DataKi:  0.0700nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479437BDBM479437(US10894807, ID P246)
Affinity DataKi:  0.160nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479444BDBM479444(US10894807, ID P253)
Affinity DataKi:  0.200nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479458BDBM479458(US10894807, ID P278)
Affinity DataKi:  0.200nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479453BDBM479453(US10894807, ID P273)
Affinity DataKi:  0.200nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479450BDBM479450(US10894807, ID P270)
Affinity DataKi:  0.200nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479415BDBM479415(US10894807, ID P200)
Affinity DataKi: <0.300nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479431BDBM479431(US10894807, ID P238)
Affinity DataKi: <0.300nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479429BDBM479429(US10894807, ID P235)
Affinity DataKi: <0.300nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479449BDBM479449(US10894807, ID P266)
Affinity DataKi:  0.300nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479442BDBM479442(US10894807, ID P251)
Affinity DataKi:  0.340nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479435BDBM479435(US10894807, ID P244)
Affinity DataKi:  0.380nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479433BDBM479433(US10894807, ID P241)
Affinity DataKi:  0.380nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479445BDBM479445(US10894807, ID P254)
Affinity DataKi:  0.400nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479457BDBM479457(US10894807, ID P277)
Affinity DataKi:  0.400nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479464BDBM479464(US10894807, ID P285)
Affinity DataKi:  0.5nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479426BDBM479426(US10894807, ID P222)
Affinity DataKi:  0.560nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479425BDBM479425(US10894807, ID P218)
Affinity DataKi:  0.600nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479438BDBM479438(US10894807, ID P247)
Affinity DataKi:  0.630nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479469BDBM479469(US10894807, ID P292)
Affinity DataKi:  0.700nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479375BDBM479375(US10894807, ID P033)
Affinity DataKi:  0.780nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479451BDBM479451(US10894807, ID P271)
Affinity DataKi:  0.800nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479463BDBM479463(US10894807, ID P283)
Affinity DataKi:  0.900nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479460BDBM479460(US10894807, ID P280)
Affinity DataKi:  0.900nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479447BDBM479447(US10894807, ID P261)
Affinity DataKi:  1nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479466BDBM479466(US10894807, ID P287)
Affinity DataKi:  1nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479462BDBM479462(US10894807, ID P282)
Affinity DataKi:  1.10nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479427BDBM479427(US10894807, ID P223)
Affinity DataKi:  1.10nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479461BDBM479461(US10894807, ID P281)
Affinity DataKi:  1.30nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479456BDBM479456(US10894807, ID P276)
Affinity DataKi:  1.30nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479448BDBM479448(US10894807, ID P263)
Affinity DataKi:  1.30nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479459BDBM479459(US10894807, ID P279)
Affinity DataKi:  1.60nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479379BDBM479379(US10894807, ID P054)
Affinity DataKi:  1.60nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479422BDBM479422(US10894807, ID P215)
Affinity DataKi:  2.20nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479452BDBM479452(US10894807, ID P272)
Affinity DataKi:  2.5nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 50246934BDBM50246934((S)-2-(3-((S)-1-carboxy-5-(4-fluorobenzamido)penty...)
Affinity DataKi:  3.10nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479421BDBM479421(US10894807, ID P212)
Affinity DataKi:  3.10nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479439BDBM479439(US10894807, ID P248)
Affinity DataKi:  3.40nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479430BDBM479430(US10894807, ID P237)
Affinity DataKi:  3.80nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479441BDBM479441(US10894807, ID P250)
Affinity DataKi:  4.10nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479468BDBM479468(US10894807, ID P291)
Affinity DataKi:  5nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479408BDBM479408(US10894807, ID P188)
Affinity DataKi:  6.60nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479455BDBM479455(US10894807, ID P275)
Affinity DataKi:  6.60nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 17659BDBM17659(pentanedioic acid analogue, (RS)-1 | 2-(phosphonom...)
Affinity DataKi:  6.60nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479419BDBM479419(US10894807, ID P204)
Affinity DataKi:  6.90nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479382BDBM479382(US10894807, ID P065)
Affinity DataKi:  9.10nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479440BDBM479440(US10894807, ID P249)
Affinity DataKi:  9.40nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479467BDBM479467(US10894807, ID P288)
Affinity DataKi:  9.70nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479376BDBM479376(US10894807, ID P045)
Affinity DataKi:  10.9nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

TargetGlutamate carboxypeptidase 2(Human)
Siemens Medical Solutions Usa

US Patent
LigandChemical structure of BindingDB Monomer ID 479381BDBM479381(US10894807, ID P059)
Affinity DataKi:  12.5nMAssay Description:The inhibitory activity of all compounds was determined using a fluorescent assay of human PSMA activity. The enzyme used in the assay was purchased ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details
US Patent

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