Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 9671
TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480719BDBM480719(US10899774, Example 35 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  1.40nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480743BDBM480743(US10899774, Example 59 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  1.60nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480754BDBM480754(US10899774, Example 70 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  2.70nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480702BDBM480702(US10899774, Example 18 | N-[rac-(2S)-2-(hydroxymet...)
Affinity DataKi:  3.40nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480707BDBM480707(US10899774, Example 23 | N-[rac-(2R)-2-(hydroxymet...)
Affinity DataKi:  3.60nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480717BDBM480717(US10899774, Example 33 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  3.70nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480720BDBM480720(US10899774, Example 36 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  3.80nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480745BDBM480745(US10899774, Example 61 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  4.60nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480721BDBM480721(US10899774, Example 37 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  5.20nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480688BDBM480688(US10899774, Example 4 | N-(2,2-dimethyl-6-morpholi...)
Affinity DataKi:  7.10nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480722BDBM480722(US10899774, Example 38 | 2-cyclopropyl-N-(2,2-dime...)
Affinity DataKi:  7.40nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480733BDBM480733(US10899774, Example 49 | 1-(2-acetamido-4-pyridyl)...)
Affinity DataKi:  7.60nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480708BDBM480708(US10899774, Example 24 | N-[rac-(2S)-2-(hydroxymet...)
Affinity DataKi:  7.70nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480744BDBM480744(US10899774, Example 60 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  8.20nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480723BDBM480723(US10899774, Example 39 | 2-bromo-N-(2,2-dimethyl-6...)
Affinity DataKi:  11nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480687BDBM480687(US10899774, Example 3 | 4-amino-N-(2,2-dimethyl-6-...)
Affinity DataKi:  13nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480750BDBM480750(US10899774, Example 66 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  14nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480747BDBM480747(US10899774, Example 63 | 6-cyano-N-[2-(hydroxymeth...)
Affinity DataKi:  16nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480718BDBM480718(US10899774, Example 34 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  17nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480746BDBM480746(US10899774, Example 62 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  17nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480735BDBM480735(US10899774, Example 51 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  18nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480716BDBM480716(US10899774, Example 32 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  19nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480741BDBM480741(US10899774, Example 57 | 6-chloro-N-[rac-(2S)-2- (...)
Affinity DataKi:  19nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480703BDBM480703(US10899774, Example 19 | N-[rac-(2R)-2-(hydroxymet...)
Affinity DataKi:  21nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480715BDBM480715(US10899774, Example 31 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  23nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480706BDBM480706(US10899774, Example 22 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  25nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480689BDBM480689(US10899774, Example 5 | 5-cyano-N-(2,2-dimethyl-6-...)
Affinity DataKi:  25nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480694BDBM480694(US10899774, Example 10 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  27nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480724BDBM480724(US10899774, Example 40 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  28nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480753BDBM480753(US10899774, Example 69 | 1-(2-cyano-4-pyridyl)-N-(...)
Affinity DataKi:  28nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480742BDBM480742(US10899774, Example 58 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  29nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480704BDBM480704(US10899774, Example 20 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  30nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480686BDBM480686(US10899774, Example 2 | N-(2,2-dimethyl-6-morpholi...)
Affinity DataKi:  30nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480710BDBM480710(US10899774, Example 26 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  35nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480709BDBM480709(US10899774, Example 25 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  35nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480699BDBM480699(US10899774, Example 15 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  36nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480740BDBM480740(US10899774, Example 56 | 6-chloro-N-[rac-(2R)-2- (...)
Affinity DataKi:  37nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480690BDBM480690(US10899774, Example 6 | N-(2,2-dimethyl-6-morpholi...)
Affinity DataKi:  38nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480711BDBM480711(US10899774, Example 27 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  42nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480725BDBM480725(US10899774, Example 41 | 2-tert-butyl-N-(2,2-dimet...)
Affinity DataKi:  43nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480691BDBM480691(US10899774, Example 7 | N-(2,2-dimethyl-6-morpholi...)
Affinity DataKi:  43nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480692BDBM480692(US10899774, Example 8 | N-(2,2-dimethyl-6-morpholi...)
Affinity DataKi:  45nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480700BDBM480700(US10899774, Example 16 | N-[rac-(2S)-2-(hydroxymet...)
Affinity DataKi:  48nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480685BDBM480685(US10899774, Example 1 | N-(2,2-dimethyl-6-morpholi...)
Affinity DataKi:  67nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480752BDBM480752(US10899774, Example 68 | 3-methyl-N-[rac-(2R)-2- (...)
Affinity DataKi:  70nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480696BDBM480696(US10899774, Example 12 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  77nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480734BDBM480734(US10899774, Example 50 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  78nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480726BDBM480726(US10899774, Example 42 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  98nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480736BDBM480736(US10899774, Example 52 | N-[2-(hydroxymethyl)-2-me...)
Affinity DataKi:  100nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

TargetInterleukin-1 receptor-associated kinase 4(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 480727BDBM480727(US10899774, Example 43 | N-(2,2-dimethyl-6-morphol...)
Affinity DataKi:  110nMAssay Description:Kinase activities were assayed using the Transcreener-Fluorecescence polarization platform (BelBrook Labs, Madison, Wis., USA) that measures amounts ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2021
Entry Details
US Patent

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