Compile Data Set for Download or QSAR
Report error Found 113 Enz. Inhib. hit(s) with all data for entry = 9725
TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484084BDBM484084(8-isopentyl-12-isopropyl-4-oxa-8,12- diazadispiro[...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484081BDBM484081(4-ethyl-9-isopentyl-1-oxa-4,9- diazaspiro[5.5]unde...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484080BDBM484080(12-ethyl-8-isopentyl-4-oxa-8,12- diazadispiro[2.1....)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484099BDBM484099(8-benzyl-12-isopropyl-4-oxa-8,12- diazadispiro[2.1...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484098BDBM484098((R)-9-benzyl-4-ethyl-2-methyl-1-oxa- 4,9-diazaspir...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484097BDBM484097(8-benzyl-12-methyl-4-oxa-8,12- diazadispiro[2.1.5....)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484096BDBM484096(8-benzyl-12-ethyl-4-oxa-8,12- diazadispiro[2.1.5.3...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484095BDBM484095(12-ethyl-8-(4-fluorobenzyl)-4-oxa-8,12- diazadispi...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484094BDBM484094(4-ethyl-9-isopentyl-2,2-dimethyl-1-oxa- 4,9-diazas...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484089BDBM484089(12-isobutyl-8-isopentyl-4-oxa-8,12- diazadispiro[2...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484088BDBM484088(8-isopentyl-12-propyl-4-oxa-8,12- diazadispiro[2.1...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484086BDBM484086((S)-4-ethyl-9-isopentyl-2-methyl-1-oxa- 4,9-diazas...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484115BDBM484115(8-(2-(3-fluoropyridin-2-yl)ethyl)-12-isopropyl-4- ...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484111BDBM484111(9-benzyl-4-ethyl-2,2-dimethyl-1-oxa- 4,9-diazaspir...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484106BDBM484106(8-benzyl-12-isobutyl-4-oxa-8,12- diazadispiro[2.1....)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484105BDBM484105(8-benzyl-12-propyl-4-oxa-8,12- diazadispiro[2.1.5....)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484103BDBM484103(8-(3,4-difluorobenzyl)-12-ethyl-4-oxa-8,12- diazad...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484102BDBM484102(12-ethyl-8-(3-fluorobenzyl)-4-oxa-8,12- diazadispi...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484101BDBM484101((S)-9-benzyl-4-ethyl-2-methyl-1-oxa- 4,9-diazaspir...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484128BDBM484128(9-isopentyl-4-propyl-1-oxa- 4,9-diazaspiro[5.5]und...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484127BDBM484127(9-(3,3-dimethylbutyl)-4- propyl-1-oxa-4,9- diazasp...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484126BDBM484126(12-isobutyl-8-(2-(6- methoxypyridin-2-yl)ethyl)-4-...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484125BDBM484125(8-(2,5-difluorophenethyl)-12- isobutyl-4-oxa-8,12-...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484124BDBM484124(9-isopentyl-4-isopropyl-2,2- dimethyl-1-oxa-4,9- d...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484121BDBM484121(8-(2-(3-fluoropyridin-2-yl)ethyl)-12-isobutyl-4- o...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484119BDBM484119(8-(2-(3-fluoropyridin-2-yl)ethyl)-12-propyl-4- oxa...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484117BDBM484117((S)-9-(2-(3-fluoropyridin-2-yl)ethyl-4-isopropyl- ...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484148BDBM484148((S)-9-(4-fluorobenzyl)-4- isopropyl-2-methyl-1-oxa...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484147BDBM484147(4-ethyl-9-(4-fluorobenzyl)- 2,2-dimethyl-1-oxa-4,9...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484146BDBM484146(8-(4-fluorobenzyl)-12-methyl- 4-oxa-8,12- diazadis...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484134BDBM484134((S)-9-isopentyl-2-methyl-4- propyl-1-oxa-4,9- diaz...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484133BDBM484133(9-isopentyl-2,2-dimethyl-4- propyl-1-oxa-4.9- diaz...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484164BDBM484164((S)-4-cyclopropyl-9-(4- fluorobenzyl)-2-methyl-1-o...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484163BDBM484163((R)-9-(4-fluorobenzyl)-2,4- dimethyl-1-oxa-4,9- di...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484162BDBM484162((S)-4-((4-isopropyl-2-methyl- 3-oxo-1-oxa-4,9- dia...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484160BDBM484160((S)-4-((4-ethyl-2-methyl-3- oxo-1-oxa-4,9- diazasp...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484156BDBM484156(4-((4-ethyl-2,2-dimethyl-3- oxo-1-oxa-4,9- diazasp...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484155BDBM484155(9-(4-chlorobenzyl)-4-ethyl- 2,2-dimethyl-1-oxa-4,9...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484154BDBM484154((R)-4-ethyl-9-(4- methoxybenzyl)-2-methyl-1- oxa-4...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484153BDBM484153((R)-4-((4-ethyl-2-methyl-3- oxo-1-oxa-4,9- diazasp...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484152BDBM484152((R)-9-(4-chlorobenzyl)-4- ethyl-2-methyl-1-oxa-4,9...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484151BDBM484151((S)-9-(4-chlorobenzyl)-4- ethyl-2-methyl-1-oxa-4,9...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484149BDBM484149((R)-4-ethyl-9-(4- fluorobenzyl)-2-methyl-1-oxa- 4,...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484180BDBM484180(8-(2-(3-chloropyridin-2- yl)ethyl)-12-isobutyl-4-o...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484168BDBM484168((S)-9-(4-fluorobenzyl)-2,4- dimethyl-1-oxa-4,9- di...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484167BDBM484167((S)-4-((2,4-dimethyl-3-oxo-1- oxa-4,9- diazaspiro[...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484166BDBM484166((S)-4-((4-cyclopropyl-2- methyl-3-oxo-1-oxa-4,9- d...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484165BDBM484165((S)-9-benzyl-4-cyclopropyl-2- methyl-1-oxa-4,9- di...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484192BDBM484192(4-isopropyl-2,2-dimethyl-9- phenethyl-1-oxa-4,9- d...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

TargetAP-4 complex subunit sigma-1(Human)
Esteve Pharmaceuticals.

US Patent
LigandChemical structure of BindingDB Monomer ID 484191BDBM484191(4-Ethyl-2-methyl-9- phenethyl-1-oxa-4,9- diazaspir...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human Sigma-1 receptor, transfected HEK-293 membranes and [3H](+)-pentazocine (Perkin Elmer, N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/6/2021
Entry Details
US Patent

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