Compile Data Set for Download or QSAR
Report error Found 228 Enz. Inhib. hit(s) with all data for entry = 9819
TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490870BDBM490870(US10975037, Example 67 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.0390nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490853BDBM490853(US10975037, Example 50 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.100nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490816BDBM490816(US10975037, Example 15 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.130nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490890BDBM490890(US10975037, Example 87 | 5-(2-(Difluoromethoxy)-4-...)
Affinity DataKd:  0.140nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490815BDBM490815(US10975037, Example 14 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.140nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490922BDBM490922(US10975037, Example 116 | 4-Chloro-5-(2-(difluorom...)
Affinity DataKd:  0.150nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490954BDBM490954(US10975037, Example 148 | 4-Chloro-5-(2-(difluorom...)
Affinity DataKd:  0.160nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490803BDBM490803(US10975037, Example 2 | 4-Chloro-5-(2-(difluoromet...)
Affinity DataKd:  0.160nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490889BDBM490889(US10975037, Example 86 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.170nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490815BDBM490815(US10975037, Example 14 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.190nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490939BDBM490939(US10975037, Example 134 | 4-Chloro-N-(((1s*,4s*)-1...)
Affinity DataKd:  0.200nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490938BDBM490938(US10975037, Example 133 | 4-Chloro-5-(2-(difluorom...)
Affinity DataKd:  0.200nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490845BDBM490845(US10975037, Example 43 | 4-Chloro-5-(2-methoxy-4-(...)
Affinity DataKd:  0.210nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490898BDBM490898(US10975037, Example 94 | Ethyl (1s*,4S*)-1-((4-chl...)
Affinity DataKd:  0.220nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490874BDBM490874(US10975037, Example 71 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.230nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490892BDBM490892(US10975037, Example 89 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.240nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490894BDBM490894(US10975037, Example 91 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.240nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490854BDBM490854(US10975037, Example 51 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.25nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490923BDBM490923(US10975037, Example 117 | 4-Chloro-5-(2-(difluorom...)
Affinity DataKd:  0.270nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490843BDBM490843(US10975037, Example 41 | 4-Chloro-5-(2-methoxy-4-(...)
Affinity DataKd:  0.280nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490999BDBM490999(US10975037, Example 193 | 4-Chloro-1-ethyl-5-(2-(m...)
Affinity DataKd:  0.280nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490879BDBM490879(US10975037, Example 76 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.280nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490875BDBM490875(US10975037, Example 72 | 4-Chloro-1-ethyl-5-(4-iso...)
Affinity DataKd:  0.290nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490872BDBM490872(US10975037, Example 69 | N-(((1r,4r)-4-(N-Carbamoy...)
Affinity DataKd:  0.290nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490846BDBM490846(US10975037, Example 44 | 4-Chloro-1-ethyl-5-(2-met...)
Affinity DataKd:  0.330nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490877BDBM490877(US10975037, Example 74 | 4-Chloro-1-ethyl-5-(4-iso...)
Affinity DataKd:  0.330nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490961BDBM490961(US10975037, Example 155 | 4-Chloro-5-(2-(difluorom...)
Affinity DataKd:  0.330nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490858BDBM490858(US10975037, Example 55 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.350nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490822BDBM490822(US10975037, Example 21 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.370nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490850BDBM490850(US10975037, Example 47 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.370nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490949BDBM490949(US10975037, Example 143 | 5-(2-(Difluoromethoxy)-4...)
Affinity DataKd:  0.370nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490849BDBM490849(US10975037, Example 46 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.420nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490844BDBM490844(US10975037, Example 42 | 4-Chloro-N-(((1s,4S)-1-hy...)
Affinity DataKd:  0.420nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490888BDBM490888(US10975037, Example 85 | 4-Chloro-1-ethyl-N-(((1s,...)
Affinity DataKd:  0.430nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490998BDBM490998(US10975037, Example 192 | 4-Chloro-1-ethyl-N-(((1s...)
Affinity DataKd:  0.430nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490823BDBM490823(US10975037, Example 22 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.440nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490971BDBM490971(US10975037, Example 165 | 4-Chloro-5-(2-chloro-4-(...)
Affinity DataKd:  0.450nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490937BDBM490937(US10975037, Example 132 | 4-Chloro-5-(2-(difluorom...)
Affinity DataKd:  0.450nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490940BDBM490940(US10975037, Example 135 | 4-Chloro-5-(2-(difluorom...)
Affinity DataKd:  0.460nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490968BDBM490968(US10975037, Example 162 | 4-Chloro-1-ethyl-N-(((1r...)
Affinity DataKd:  0.480nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490970BDBM490970(US10975037, Example 164 | 4-Chloro-5-(2-chloro-4-(...)
Affinity DataKd:  0.5nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490893BDBM490893(US10975037, Example 90 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.510nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490848BDBM490848(US10975037, Example 45 | 4-Chloro-1-ethyl-N-(((1s,...)
Affinity DataKd:  0.570nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490944BDBM490944(US10975037, Example 139 | 4-Chloro-5-(2-(difluorom...)
Affinity DataKd:  0.580nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490881BDBM490881(US10975037, Example 78 | 5-(2-(Difluoromethoxy)-4-...)
Affinity DataKd:  0.590nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490802BDBM490802(US10975037, Example 1 | Step b | 4-Chloro-1-ethyl-...)
Affinity DataKd:  0.600nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490876BDBM490876(US10975037, Example 73 | 4-Chloro-1-ethyl-N-(((1s,...)
Affinity DataKd:  0.630nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490804BDBM490804(US10975037, Example 3 | 4-Chloro-1-ethyl-5-(2-meth...)
Affinity DataKd:  0.630nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490969BDBM490969(US10975037, Example 163 | 4-Chloro-1-ethyl-N-(((1s...)
Affinity DataKd:  0.630nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

TargetNuclear receptor ROR-gamma(Human)
Janssen Pharmaceutica

US Patent
LigandChemical structure of BindingDB Monomer ID 490857BDBM490857(US10975037, Example 54 | 4-Chloro-5-(2-(difluorome...)
Affinity DataKd:  0.690nMAssay Description:ThermoFluor experiments were carried out using instruments owned by Janssen Research and Development, L.L.C. through its acquisition of 3-Dimensional...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2021
Entry Details
US Patent

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