Compile Data Set for Download or QSAR
Report error Found 217 Enz. Inhib. hit(s) with all data for entry = 9990
TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505120BDBM505120(US11066409, Compound I-0003)
Affinity DataIC50: 1.80nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505144BDBM505144(US11066409, Compound I-0188)
Affinity DataIC50: 7.60nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505150BDBM505150(US11066409, Compound I-0007)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505213BDBM505213(US11066409, Compound I-0074)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505151BDBM505151(US11066409, Compound I-0008)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505152BDBM505152(US11066409, Compound I-0010)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505153BDBM505153(US11066409, Compound I-0011)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505216BDBM505216(US11066409, Compound I-0077)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505154BDBM505154(US11066409, Compound I-0012)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505155BDBM505155(US11066409, Compound I-0013)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505156BDBM505156(US11066409, Compound I-0014)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505219BDBM505219(US11066409, Compound I-0080)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505161BDBM505161(US11066409, Compound I-0019)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505162BDBM505162(US11066409, Compound I-0020)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505199BDBM505199(US11066409, Compound I-0058)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505262BDBM505262(US11066409, Compound I-0134 | US11066409, Compound...)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505205BDBM505205(US11066409, Compound I-0065)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505206BDBM505206(US11066409, Compound I-0066)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505207BDBM505207(US11066409, Compound I-0067)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505147BDBM505147(US11066409, Compound I-0002)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505180BDBM505180(US11066409, Compound I-0039)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505240BDBM505240(US11066409, Compound I-0110 | US11066409, Compound...)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505182BDBM505182(US11066409, Compound I-0041)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505130BDBM505130(US11066409, Compound I-0111 | US11066409, Compound...)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505183BDBM505183(US11066409, Compound I-0042)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505184BDBM505184(US11066409, Compound I-0043)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505125BDBM505125(US11066409, Compound I-0069)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505190BDBM505190(US11066409, Compound I-0049)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505191BDBM505191(US11066409, Compound I-0050)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505195BDBM505195(US11066409, Compound I-0054)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505164BDBM505164(US11066409, Compound I-0022)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505165BDBM505165(US11066409, Compound I-0023)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505168BDBM505168(US11066409, Compound I-0026)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505169BDBM505169(US11066409, Compound I-0027)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505170BDBM505170(US11066409, Compound I-0028)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505171BDBM505171(US11066409, Compound I-0029)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505235BDBM505235(US11066409, Compound I-0097)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505236BDBM505236(US11066409, Compound I-0098)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505237BDBM505237(US11066409, Compound I-0099)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505178BDBM505178(US11066409, Compound I-0037)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505179BDBM505179(US11066409, Compound I-0038)
Affinity DataIC50: 10nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505124BDBM505124(US11066409, Compound I-0059)
Affinity DataIC50: 11nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505128BDBM505128(US11066409, Compound I-0102)
Affinity DataIC50: 11nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505129BDBM505129(US11066409, Compound I-0106)
Affinity DataIC50: 11nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505127BDBM505127(US11066409, Compound I-0100)
Affinity DataIC50: 12nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505135BDBM505135(US11066409, Compound I-0151)
Affinity DataIC50: 14nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505119BDBM505119(US11066409, Compound I-0001)
Affinity DataIC50: 16nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505123BDBM505123(US11066409, Compound I-0032)
Affinity DataIC50: 16nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505136BDBM505136(US11066409, Compound I-0154)
Affinity DataIC50: 17nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

TargetP2X purinoceptor 7(Human)
Shionogi

US Patent
LigandChemical structure of BindingDB Monomer ID 505126BDBM505126(US11066409, Compound I-0091)
Affinity DataIC50: 17nMAssay Description:Evaluation of a human P2X7 receptor inhibitory activity Stably expressing cell line (1321N1 cell transfected with the human P2X7 receptor gene (GenBa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2021
Entry Details
US Patent

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