Compile Data Set for Download or QSAR
Report error Found 367 Enz. Inhib. hit(s) with all data for entry = 10028
TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192311BDBM192311(US9670204, 105 1-(2-((2-ethyl-6-(1-(methylsulfonyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 426470BDBM426470(US10526329, Compound 106 | US10526329, Compound 10...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192363BDBM192363(US9670204, 108 ethyl2-(4-(2-ethyl-3-((4-(4-fluorop...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192475BDBM192475(US9670204, 109 ethyl2-(4-(2-ethyl-3-((4-(4-fluorop...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192476BDBM192476(US9670204, 110 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192576BDBM192576(US9670204, 111 (R)-2-(4-(2-ethyl-3-((4-(4-fluoroph...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192613BDBM192613(US9670204, 112 (S)-2-(4-(2-ethyl-3-((4-(4-fluoroph...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192614BDBM192614(US9670204, 113 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192615BDBM192615(US9670204, 114 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192616BDBM192616(US9670204, 115 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 426480BDBM426480(US10526329, Compound 116 | US11072611, Compound 11...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192775BDBM192775(US9670204, 118 4-((4-(2-ethyl-3-((4-(4-fluoropheny...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192788BDBM192788(US9670204, 124 1-(3,3-difluoroazetidin-1-yl)-2-(4-...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192790BDBM192790(US9670204, 125 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192791BDBM192791(US9670204, 126 1-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192914BDBM192914(US9670204, 128 1-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 191618BDBM191618(US9670204, 22 2-(4-(3-((5-cyano-4-(4-fluorophenyl)...)
Affinity DataIC50: 50nMAssay Description:TABLE V: 5 μL of a dilution series of compound, starting from 20 μM highest concentration, 1/5 dilution, is added to the wells. hENPP2 is u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192189BDBM192189(US9670204, 86 N-(6-(1-(3-chloropropylsulfonyl)pipe...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192190BDBM192190(US9670204, 87 N-(6-(1-(3-(dimethylamino)propyl-sul...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192192BDBM192192(US9670204, 88 N-(2-ethyl-6-(1-(3-morpholinopropyl-...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192212BDBM192212(US9670204, 89 N-(2-ethyl-6-(1-(3-(pyrrolidin-1-yl)...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192214BDBM192214(US9670204, 90 N-(6-(1-(3-aminopropylsulfonyl)piper...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192215BDBM192215(US9670204, 91 N-(2-ethyl-6-(1-(2-morpholinoethylsu...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192218BDBM192218(US9670204, 92 4-(2-ethyl-3-((4-(4-fluorophenyl)thi...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192219BDBM192219(US9670204, 93 3-(4-(2-ethyl-3-((4-(4-fluorophenyl)...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 191784BDBM191784(US9670204, 30 1-(azetidin-1-yl)-2-(4-(2-ethyl-3-((...)
Affinity DataIC50: 50nMAssay Description:TABLE V: 5 μL of a dilution series of compound, starting from 20 μM highest concentration, 1/5 dilution, is added to the wells. hENPP2 is u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 191872BDBM191872(US9670204, 74 3-(4-(2-ethyl-3-((4-(4-fluorophenyl)...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 191788BDBM191788(US9670204, 31 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)...)
Affinity DataIC50: 50nMAssay Description:TABLE V: 5 μL of a dilution series of compound, starting from 20 μM highest concentration, 1/5 dilution, is added to the wells. hENPP2 is u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192253BDBM192253(US9670204, 94 3-(4-(2-ethyl-3-((4-(4-fluorophenyl)...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192268BDBM192268(US9670204, 96 2-(2-((2-ethyl-6-(1-(methylsulfonyl)...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192286BDBM192286(US9670204, 98 N-(2-ethyl-6-(1-(methylsulfonyl)pipe...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192288BDBM192288(US9670204, 99 4-(2-chloro-4-fluorophenyl)-N-(2-eth...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192291BDBM192291(US9670204, 100 4-(2,4-difluorophenyl)-N-(2-ethyl-6...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192297BDBM192297(US9670204, 103 4-(4-fluorophenyl)-N-(2-ethyl-6-(1-...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192172BDBM192172(US9670204, 80 N-(2-ethyl-6-(1-(methylsulfonyl)pipe...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192982BDBM192982(US9670204, 162 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyaz...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192986BDBM192986(US9670204, 166 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyaz...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192987BDBM192987(US9670204, 167 2-(2-((6-(4-(2-(azetidin-1-yl)-2-ox...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192988BDBM192988(US9670204, 168 2-(4-(3-((4-(2-cyano-4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192990BDBM192990(US9670204, 170 2-(2-((2-ethyl-6-(1-(2-(3-hydroxyaz...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192991BDBM192991(US9670204, 171 2-(4-(3-((4-(2-cyano-4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192992BDBM192992(US9670204, 172 2-(2-((2-ethyl-6-(1-(2-(3-hydroxyaz...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192993BDBM192993(US9670204, 173 2-(5-((2-ethyl-6-(1-(2-(3-hydroxyaz...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192994BDBM192994(US9670204, 174 2-(4-(2-(2-cyanoethyl)-3-((4-(4-flu...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192999BDBM192999(US9670204, 179 N-(1-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 193000BDBM193000(US9670204, 180 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 193002BDBM193002(US9670204, 182 4-(2-ethyl-3-((4-(4-fluorophenyl)th...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 193003BDBM193003(US9670204, 183 1-(3-((4-(4-chlorophenyl)thiazol-2-...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 193004BDBM193004(US9670204, 184 ethyl2-(3-(3-((4-(4-chlorophenyl)th...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 193005BDBM193005(US9670204, 185 4-(4-chlorophenyl)-N-methyl-N-(6-(1...)
Affinity DataIC50: 50nMAssay Description:TABLE VI: (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotaxin substrate FS-3 as substrate. FS-3 is a doubly l...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/7/2022
Entry Details
US Patent

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