Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 10177
LigandChemical structure of BindingDB Monomer ID 446461BDBM446461(US10669271, Example 14 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446462BDBM446462(US10669271, Example 15 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446463BDBM446463(US10669271, Example 16 | US10669271, Example 19 | ...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446464BDBM446464(US10669271, Example 17 | US10669271, Example 20 | ...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446465BDBM446465(US10669271, Example 18 | US10669271, Example 21 | ...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 518543BDBM518543(US11124511, Example 19 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 518544BDBM518544(US11124511, Example 20 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 518545BDBM518545(US11124511, Example 21 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446469BDBM446469(US10669271, Example 22 | (S)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446470BDBM446470(US10669271, Example 23 | (S)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446471BDBM446471(US10669271, Example 24 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446472BDBM446472(US10669271, Example 25 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446473BDBM446473(US10669271, Example 26 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446474BDBM446474(US10669271, Example 27 | (R)-3-(1-((7-cyano-2-(3&#...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446475BDBM446475(US10669271, Example 28 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446476BDBM446476(US10669271, Example 29 | (R)-1-((2-(3′-(2-am...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446448BDBM446448(US10669271, Example 1 | (R)-1-((7-cyano-2-(3′...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446449BDBM446449(US10669271, Example 2 | (R)-1-((7-cyano-2-(3′...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446450BDBM446450(US10669271, Example 3 | (S)-1-((7-cyano-2-(3′...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446451BDBM446451(US10669271, Example 4 | (S)-1-((7-cyano-2-(3′...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446452BDBM446452(US10669271, Example 5 | (S)-1-((7-cyano-2-(3′...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446453BDBM446453(US10669271, Example 6 | US10669271, Example 33 | (...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446454BDBM446454(US10669271, Example 7 | (R)-1-((7-cyano-2-(3′...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446454BDBM446454(US10669271, Example 7 | (R)-1-((7-cyano-2-(3′...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446456BDBM446456(US10669271, Example 9 | (R)-1-((7-cyano-2-(3′...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446457BDBM446457(US10669271, Example 10 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446458BDBM446458(US10669271, Example 11 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446459BDBM446459(US10669271, Example 12 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446460BDBM446460(US10669271, Example 13 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446477BDBM446477(US10669271, Example 30 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446478BDBM446478(US10669271, Example 31 | (S)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446479BDBM446479(US10669271, Example 32 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 518558BDBM518558(US11124511, Example 33 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 446481BDBM446481(US10669271, Example 34 | (R)-1-((7-cyano-2-(3̸...)
Affinity DataIC50: 10nMAssay Description:The assays were conducted in a standard black 384-well polystyrene plate with a final volume of 20 μL. Inhibitors were first serially diluted in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2022
Entry Details
US Patent