Compile Data Set for Download or QSAR
maximum 50k data
Found 96 Enz. Inhib. hit(s) with all data for entry = 10277
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524345((S)-2-fluoro-4-(5-(1-methyl-1H-indazol-5- yl)-1-(p...)
Affinity DataIC50:  2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524395(2-fluoro-4-(5-(1-methyl-1H-indazol-5-yl)- 1-((1-me...)
Affinity DataIC50:  2.10nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524392(4-(1-(azepan-4-ylmethyl)-5-(1-methyl-1H- indazol-5...)
Affinity DataIC50:  2.20nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524347((S)-4-(5-(1-ethyl-1H-indazol-5-yl)-1- (pyrrolidin-...)
Affinity DataIC50:  4nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524379(4-(1-(azepan-4-ylmethyl)-5-(1-methyl-1H- indazol-5...)
Affinity DataIC50:  4nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524399(4-(5-(4-methyl-3,4-dihydro-2H- benzo[b][1,4]oxazin...)
Affinity DataIC50:  4.10nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524381(4-(5-(1-methyl-1H-indazol-5-yl)-1-((1- methylazepa...)
Affinity DataIC50:  4.10nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524398(4-(5-(1-methyl-1H-indazol-5-yl)-1-((4- methylpiper...)
Affinity DataIC50:  5.20nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524397(4-(1-((8-azabicyclo[3.2.1]octan-3- yl)methyl)-5-(1...)
Affinity DataIC50:  5.30nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524327((R)-2-fluoro-4-(5-(1-methyl-1H-indazol-5- yl)-1-(p...)
Affinity DataIC50:  6nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524346((S)-2-fluoro-4-(5-(2-methyl-2H-indazol-5- yl)-1-(p...)
Affinity DataIC50:  7nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524322((R)-2-fluoro-4-(5-(2-methyl-2H-indazol-5- yl)-1-(p...)
Affinity DataIC50:  7nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524385(4-(5-(1-methyl-1H-indol-5-yl)-1- (piperidin-4-ylme...)
Affinity DataIC50:  7.10nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524369(4-(5-(1-methyl-1H-indazol-5-yl)-1- (piperidin-4-yl...)
Affinity DataIC50:  7.60nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524340((R)-2-fluoro-4-(5-(4-methyl-3,4-dihydro- 2H-benzo[...)
Affinity DataIC50:  8nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524335((R)-4-(5-(1-ethyl-1H-indazol-5-yl)-1- (pyrrolidin-...)
Affinity DataIC50:  8nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524342(2-fluoro-4-(5-(1-methyl-1H-indazol-5-yl)- 1-(piper...)
Affinity DataIC50:  11nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524341((R)-2-fluoro-4-(5-(1-methyl-1H-indazol-5- yl)-1-(p...)
Affinity DataIC50:  11nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524375(4-(1-(4-aminobutyl)-5-(1-methyl-1H- indazol-5-yl)-...)
Affinity DataIC50:  13nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524363(2-fluoro-4-(5-(1-methyl-1H-indazol-5-yl)- 1-((1-me...)
Affinity DataIC50:  13.7nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524380(4-(1-((1-(2-hydroxyethyl)piperidin-4- yl)methyl)-5...)
Affinity DataIC50:  14.3nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524310((R)-2-fluoro-4-(6-(1-methyl-1H-indazol-5- yl)-3-(p...)
Affinity DataIC50:  14.6nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524396(4-(1-((2,6-dimethylpiperidin-4-yl)methyl)- 5-(1-me...)
Affinity DataIC50:  16.2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524373(2-fluoro-4-(1-((1-(2- hydroxyethyl)piperidin-4-yl)...)
Affinity DataIC50:  16.2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524319((R)-4-(5-(1-methyl-1H-indazol-5-yl)-1- (pyrrolidin...)
Affinity DataIC50:  18nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524365(4-(1-(3-aminopropyl)-5-(1-methyl-1H- indazol-5-yl)...)
Affinity DataIC50:  18.3nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524336((R)-2-fluoro-4-(5-(1-methyl-1H- benzo[d]imidazol-5...)
Affinity DataIC50:  19nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524400(4-(5-(benzo[d][1,3]dioxol-5-yl)-1- (piperidin-4-yl...)
Affinity DataIC50:  20.5nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524344(3-fluoro-4-(5-(1-methyl-1H-indazol-5-yl)- 1-(((R)-...)
Affinity DataIC50:  21nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524387(4-(5-(4-(dimethylamino)phenyl)-1- (piperidin-4-ylm...)
Affinity DataIC50:  23.1nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524316((R)-4-(5-(2-methyl-2H-indazol-5-yl)-1- (pyrrolidin...)
Affinity DataIC50:  25nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524338((R)-2-fluoro-4-(5-(2-methyl-2H-indazol-6- yl)-1-(p...)
Affinity DataIC50:  26nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524330((R)-2-fluoro-4-(5-(1-isopropyl-1H- indazol-5-yl)-1...)
Affinity DataIC50:  26nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524334((R)-4-(5-(2-ethyl-2H-indazol-5-yl)-1- (pyrrolidin-...)
Affinity DataIC50:  27nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524370(4-(5-(1-methyl-1H-indazol-5-yl)-1-((1- methylpiper...)
Affinity DataIC50:  28nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524364(4-(1-((1-ethylpiperidin-4-yl)methyl)-5-(1- methyl-...)
Affinity DataIC50:  28.2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524372(2-fluoro-4-(1-((4-hydroxy-1- methylpiperidin-4-yl)...)
Affinity DataIC50:  28.4nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524374(4-(1-(3-aminopropyl)-5-(1-methyl-1H- indazol-5-yl)...)
Affinity DataIC50:  28.5nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524377(4-(1-((1-ethylpiperidin-4-yl)methyl)-5-(1- methyl-...)
Affinity DataIC50:  30.2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524378((R)-4-(5-(1-methyl-1H-indazol-5-yl)-1- ((1-methylp...)
Affinity DataIC50:  32.7nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524389(4-(5-(4-(dimethylamino)phenyl)-1-((1- methylpiperi...)
Affinity DataIC50:  34.6nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524390(3-fluoro-4-(5-(1-methyl-1H-indazol-5-yl)- 1-(piper...)
Affinity DataIC50:  38.1nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524376(4-(5-(1-methyl-1H-indazol-5-yl)-1-(3- (methylamino...)
Affinity DataIC50:  39.4nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524339((R)-4-(5-(4-(3,5-dimethyl-1H-pyrazol-1- yl)phenyl)...)
Affinity DataIC50:  40nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524352((R)-2-fluoro-4-(5-(1-methyl-1H-indazol-5- yl)-1-((...)
Affinity DataIC50:  42nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524307((R)-2-fluoro-4-(5-(2-methyl-2H-indazol-5- yl)-1-(p...)
Affinity DataIC50:  49nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524324(4-(5-(2-methyl-2H-indazol-5-yl)-1- (piperidin-4-yl...)
Affinity DataIC50:  51nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524318((R)-N-(4-(4-(4-cyanophenyl)-1- (pyrrolidin-3-ylmet...)
Affinity DataIC50:  52nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524331((R)-2-fluoro-4-(5-(2-isopropyl-2H- indazol-5-yl)-1...)
Affinity DataIC50:  60nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM524348((R)-4-(5-(1,3-dimethyl-1H-indazol-5-yl)- 1-(pyrrol...)
Affinity DataIC50:  61nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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