Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with all data for entry = 10277
TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524345BDBM524345(US11168082, Cpd. No. 41 | (S)-2-fluoro-4-(5-(1-met...)
Affinity DataIC50: 2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524395BDBM524395(US11168082, Cpd. No. 94 | 2-fluoro-4-(5-(1-methyl-...)
Affinity DataIC50: 2.10nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524392BDBM524392(US11168082, Cpd. No. 91 | 4-(1-(azepan-4-ylmethyl)...)
Affinity DataIC50: 2.20nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524347BDBM524347(US11168082, Cpd. No. 43 | (S)-4-(5-(1-ethyl-1H-ind...)
Affinity DataIC50: 4nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524379BDBM524379(US11168082, Cpd. No. 77 | 4-(1-(azepan-4-ylmethyl)...)
Affinity DataIC50: 4nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524381BDBM524381(US11168082, Cpd. No. 79 | 4-(5-(1-methyl-1H-indazo...)
Affinity DataIC50: 4.10nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524399BDBM524399(US11168082, Cpd. No. 98 | 4-(5-(4-methyl-3,4-dihyd...)
Affinity DataIC50: 4.10nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524398BDBM524398(US11168082, Cpd. No. 97 | 4-(5-(1-methyl-1H-indazo...)
Affinity DataIC50: 5.20nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524397BDBM524397(US11168082, Cpd. No. 96 | 4-(1-((8-azabicyclo[3.2....)
Affinity DataIC50: 5.30nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524327BDBM524327(US11168082, Cpd. No. 23 | (R)-2-fluoro-4-(5-(1-met...)
Affinity DataIC50: 6nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524322BDBM524322(US11168082, Cpd. No. 18 | (R)-2-fluoro-4-(5-(2-met...)
Affinity DataIC50: 7nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524346BDBM524346(US11168082, Cpd. No. 42 | (S)-2-fluoro-4-(5-(2-met...)
Affinity DataIC50: 7nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524385BDBM524385(US11168082, Cpd. No. 83 | 4-(5-(1-methyl-1H-indol-...)
Affinity DataIC50: 7.10nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524369BDBM524369(US11168082, Cpd. No. 67 | 4-(5-(1-methyl-1H-indazo...)
Affinity DataIC50: 7.60nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524340BDBM524340(US11168082, Cpd. No. 36 | (R)-2-fluoro-4-(5-(4-met...)
Affinity DataIC50: 8nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524335BDBM524335(US11168082, Cpd. No. 31 | (R)-4-(5-(1-ethyl-1H-ind...)
Affinity DataIC50: 8nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524341BDBM524341(US11168082, Cpd. No. 37 | (R)-2-fluoro-4-(5-(1-met...)
Affinity DataIC50: 11nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524342BDBM524342(US11168082, Cpd. No. 38 | 2-fluoro-4-(5-(1-methyl-...)
Affinity DataIC50: 11nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524375BDBM524375(US11168082, Cpd. No. 73 | 4-(1-(4-aminobutyl)-5-(1...)
Affinity DataIC50: 13nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524363BDBM524363(US11168082, Cpd. No. 60 | 2-fluoro-4-(5-(1-methyl-...)
Affinity DataIC50: 13.7nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524380BDBM524380(US11168082, Cpd. No. 78 | 4-(1-((1-(2-hydroxyethyl...)
Affinity DataIC50: 14.3nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524310BDBM524310(US11168082, Cpd. No. 6 | (R)-2-fluoro-4-(6-(1-meth...)
Affinity DataIC50: 14.6nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524373BDBM524373(US11168082, Cpd. No. 71 | 2-fluoro-4-(1-((1-(2- hy...)
Affinity DataIC50: 16.2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524396BDBM524396(US11168082, Cpd. No. 95 | 4-(1-((2,6-dimethylpiper...)
Affinity DataIC50: 16.2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524319BDBM524319(US11168082, Cpd. No. 15 | (R)-4-(5-(1-methyl-1H-in...)
Affinity DataIC50: 18nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524365BDBM524365(US11168082, Cpd. No. 62 | 4-(1-(3-aminopropyl)-5-(...)
Affinity DataIC50: 18.3nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524336BDBM524336(US11168082, Cpd. No. 32 | (R)-2-fluoro-4-(5-(1-met...)
Affinity DataIC50: 19nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524400BDBM524400(US11168082, Cpd. No. 99 | 4-(5-(benzo[d][1,3]dioxo...)
Affinity DataIC50: 20.5nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524344BDBM524344(US11168082, Cpd. No. 40 | 3-fluoro-4-(5-(1-methyl-...)
Affinity DataIC50: 21nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524387BDBM524387(US11168082, Cpd. No. 85 | 4-(5-(4-(dimethylamino)p...)
Affinity DataIC50: 23.1nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524316BDBM524316(US11168082, Cpd. No. 12 | (R)-4-(5-(2-methyl-2H-in...)
Affinity DataIC50: 25nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524338BDBM524338(US11168082, Cpd. No. 34 | (R)-2-fluoro-4-(5-(2-met...)
Affinity DataIC50: 26nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524330BDBM524330(US11168082, Cpd. No. 26 | (R)-2-fluoro-4-(5-(1-iso...)
Affinity DataIC50: 26nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524334BDBM524334(US11168082, Cpd. No. 30 | (R)-4-(5-(2-ethyl-2H-ind...)
Affinity DataIC50: 27nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524370BDBM524370(US11168082, Cpd. No. 68 | 4-(5-(1-methyl-1H-indazo...)
Affinity DataIC50: 28nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524364BDBM524364(US11168082, Cpd. No. 61 | 4-(1-((1-ethylpiperidin-...)
Affinity DataIC50: 28.2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524372BDBM524372(US11168082, Cpd. No. 70 | 2-fluoro-4-(1-((4-hydrox...)
Affinity DataIC50: 28.4nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524374BDBM524374(US11168082, Cpd. No. 72 | 4-(1-(3-aminopropyl)-5-(...)
Affinity DataIC50: 28.5nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524377BDBM524377(US11168082, Cpd. No. 75 | 4-(1-((1-ethylpiperidin-...)
Affinity DataIC50: 30.2nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524378BDBM524378(US11168082, Cpd. No. 76 | (R)-4-(5-(1-methyl-1H-in...)
Affinity DataIC50: 32.7nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524389BDBM524389(US11168082, Cpd. No. 87 | 4-(5-(4-(dimethylamino)p...)
Affinity DataIC50: 34.6nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524390BDBM524390(US11168082, Cpd. No. 89 | 3-fluoro-4-(5-(1-methyl-...)
Affinity DataIC50: 38.1nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524376BDBM524376(US11168082, Cpd. No. 74 | 4-(5-(1-methyl-1H-indazo...)
Affinity DataIC50: 39.4nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524339BDBM524339(US11168082, Cpd. No. 35 | (R)-4-(5-(4-(3,5-dimethy...)
Affinity DataIC50: 40nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524352BDBM524352(US11168082, Cpd. No. 49 | (R)-2-fluoro-4-(5-(1-met...)
Affinity DataIC50: 42nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524307BDBM524307(US11168082, Cpd. No. 3 | (R)-2-fluoro-4-(5-(2-meth...)
Affinity DataIC50: 49nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524324BDBM524324(US11168082, Cpd. No. 20 | 4-(5-(2-methyl-2H-indazo...)
Affinity DataIC50: 51nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524318BDBM524318(US11168082, Cpd. No. 14 | (R)-N-(4-(4-(4-cyanophen...)
Affinity DataIC50: 52nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524331BDBM524331(US11168082, Cpd. No. 27 | (R)-2-fluoro-4-(5-(2-iso...)
Affinity DataIC50: 60nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 524348BDBM524348(US11168082, Cpd. No. 44 | (R)-4-(5-(1,3-dimethyl-1...)
Affinity DataIC50: 61nMAssay Description:Human recombinant LSD1 protein expressed in E. coli cells was purchased from Active Motif (Carlsbad, Calif.). Biotin-labeled Histone H3K4Me peptide (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details
US Patent

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