Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 10310
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shenzhen Targetrx

US Patent
LigandPNGBDBM526931((S)-1-(3-(4-amino-5-(4-phenoxyphenyl)-5H-pyrrolo[3...)
Affinity DataIC50: <1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shenzhen Targetrx

US Patent
LigandPNGBDBM526932((R)-1-(3-(4-amino-5-(4-phenoxyphenyl)-5H-pyrrolo[3...)
Affinity DataIC50: <1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shenzhen Targetrx

US Patent
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50: <1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shenzhen Targetrx

US Patent
LigandPNGBDBM526934((S)-1-(3-(7-amino-1-(4-phenoxyphenyl)-1H-pyrazolo[...)
Affinity DataIC50: <1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shenzhen Targetrx

US Patent
LigandPNGBDBM526935((S)-1-(3-(8-amino-1-(4-phenoxyphenyl)-1H-pyrazolo[...)
Affinity DataIC50: <1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Shenzhen Targetrx

US Patent
LigandPNGBDBM526933((R)-1-(3-(7-amino-1-(4-phenoxyphenyl)-1H-pyrazolo[...)
Affinity DataIC50: <1nMAssay Description:BTK (Invitrogen, catalog number: PR5442A), HTRF-TK kit (Cisbio, catalog number: 62TK0PEC), MgCl2 (SIGMA, catalog number: 63020-1L), ATP (Sigma, catal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent