Compile Data Set for Download or QSAR
Report error Found 49 Enz. Inhib. hit(s) with all data for entry = 10332
LigandChemical structure of BindingDB Monomer ID 528485BDBM528485(US11191765, Example 37 | 5-(3,4-Dimethoxyphenyl)-[...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528484BDBM528484(US11191765, Example 36 | 2-(2-Chlorophenyl)-5-phen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528487BDBM528487(US11191765, Example 1 | 5-(Benzo[d][1,3]dioxol-5-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528486BDBM528486(US11191765, Example 38 | 5-(4-Methoxyphenyl)-[1,2,...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528489BDBM528489(US11191765, Example 3 | 5-(1H-Indazol-5-yl)-2-(pyr...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528488BDBM528488(US11191765, Example 2 | 5-(1H-Benzo[d][1,2,3]triaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528491BDBM528491(US11191765, Example 5 | 2-Ethyl-5-(1H-indazol-5-yl...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528490BDBM528490(US11191765, Example 4 | 5-(1H-indazol-5-yl)-2-meth...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528493BDBM528493(US11191765, Example 7 | 5-(1H-Benzo[d][1,2,3]triaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528492BDBM528492(US11191765, Example 6 | 5-(1H-Benzo[d][1,2,3]triaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528476BDBM528476(US11191765, Example 9 | 5-(4-Chloro-3-methoxypheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528405BDBM528405(US11191765, Example 8 | 5-(4-Chloro-3-methoxypheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528495BDBM528495(US11191765, Example 11 | 5-(1H-Benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528494BDBM528494(US11191765, Example 10 | 2-(3,4-Dichlorophenyl)-5-...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528497BDBM528497(US11191765, Example 13 | 5-(1H-Benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528496BDBM528496(US11191765, Example 12 | 2-(3-Chlorophenyl)-5-(1H-...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528405BDBM528405(US11191765, Example 8 | 5-(4-Chloro-3-methoxypheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528477BDBM528477(US11191765, Example 15 | 5-(Benzo[d][1,3]dioxol-5-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528476BDBM528476(US11191765, Example 9 | 5-(4-Chloro-3-methoxypheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528479BDBM528479(US11191765, Example 31 | 2,5-Diphenyl-[1,2,4]triaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528478BDBM528478(US11191765, Example 30 | 5-(2-Methoxyphenyl)-2-phe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528481BDBM528481(US11191765, Example 33 | 5-(3-Methoxyphenyl)-2-phe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528480BDBM528480(US11191765, Example 32 | 5-(4-Methoxyphenyl)-2-phe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528483BDBM528483(US11191765, Example 35 | 2-(4-Methoxyphenyl)-5-phe...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528482BDBM528482(US11191765, Example 34 | 2-(4-Chlorophenyl)-5-(4-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:Purified PASK (UniProt #Q96RG2; human recombinant N-terminal GST tagged construct, residues 879-1323) from insect cells (final concentration 5 nM) is...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528513BDBM528513(US11191765, Example 39 | 5-(1H-Benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528482BDBM528482(US11191765, Example 34 | 2-(4-Chlorophenyl)-5-(4-m...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528515BDBM528515(US11191765, Example 41 | 5-(1H-Benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528514BDBM528514(US11191765, Example 40 | 5-(1H-Benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528517BDBM528517(US11191765, Example 43 | 5-(1H-Benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528516BDBM528516(US11191765, Example 42 | 2-(4-Chlorophenyl)-5-(1-e...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528519BDBM528519(US11191765, Example 45 | 5-(1H-Benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528518BDBM528518(US11191765, Example 44 | 2-(4-Chlorophenyl)-5-(1H-...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528477BDBM528477(US11191765, Example 15 | 5-(Benzo[d][1,3]dioxol-5-...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528498BDBM528498(US11191765, Example 14 | 5-(1H-Benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528500BDBM528500(US11191765, Example 17 | 5-(2,3-Dihydrobenzo[b][1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528499BDBM528499(US11191765, Example 16 | 5-(2,3-Dihydrobenzo[b][1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528502BDBM528502(US11191765, Example 19 | 2-Benzyl-5-(4-methoxyphen...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528501BDBM528501(US11191765, Example 18 | 2-Benzyl-5-(2,3-dihydrobe...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528504BDBM528504(US11191765, Example 21 | 5-(1-Ethyl-1H-indazol-5-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528503BDBM528503(US11191765, Example 20 | 2-(4-Fluorophenyl)-5-(1H-...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528506BDBM528506(US11191765, Example 23 | 5-(1H-benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528505BDBM528505(US11191765, Example 22 | 5-(1H-Benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528508BDBM528508(US11191765, Example 25)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528507BDBM528507(US11191765, Example 24 | 5-(1H-benzo[d][1,2,3]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528510BDBM528510(US11191765, Example 27 | 5-(4-Methoxyphenyl)-2-met...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528486BDBM528486(US11191765, Example 38 | 5-(4-Methoxyphenyl)-[1,2,...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528512BDBM528512(US11191765, Example 29 | 5-(Benzo[d][1,3]dioxol-5-...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 528511BDBM528511(US11191765, Example 28 | 5-(2,3-Dihydrobenzo[b][1,...)
Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2022
Entry Details
US Patent