Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 10398
TargetProtein O-GlcNAcase(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 532950BDBM532950(US11214576, Example 2 | (-)-5-fluoro-6-[1-[4-(5-me...)
Affinity DataIC50: 1.13nMAssay Description:The assay buffer is prepared to give a final concentration of 50 mM H2NaPO3 HNa2PO3, 0.01% bovine serum albumin and 0.01% Triton X-100 in water, at p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2022
Entry Details
US Patent

TargetProtein O-GlcNAcase(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 532948BDBM532948(US11214576, Example 1 | (-)-6-[1-[4-(5-methyl-1,3,...)
Affinity DataIC50: 1.24nMAssay Description:The assay buffer is prepared to give a final concentration of 50 mM H2NaPO3 HNa2PO3, 0.01% bovine serum albumin and 0.01% Triton X-100 in water, at p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2022
Entry Details
US Patent

TargetProtein O-GlcNAcase(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 532951BDBM532951(US11214576, Example 3 | (+)-6-[(1R)-1-[4-(5-methyl...)
Affinity DataIC50: 611nMAssay Description:The assay buffer is prepared to give a final concentration of 50 mM H2NaPO3 HNa2PO3, 0.01% bovine serum albumin and 0.01% Triton X-100 in water, at p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2022
Entry Details
US Patent

TargetProtein O-GlcNAcase(Human)
Eli Lilly

US Patent
LigandChemical structure of BindingDB Monomer ID 532952BDBM532952(US11214576, Example 4 | (+)-5-fluoro-6-[1-[4-(5-me...)
Affinity DataIC50: 2.66E+3nMAssay Description:The assay buffer is prepared to give a final concentration of 50 mM H2NaPO3 HNa2PO3, 0.01% bovine serum albumin and 0.01% Triton X-100 in water, at p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/8/2022
Entry Details
US Patent