Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 10405
TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533383BDBM533383(US11220510, Example 20)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533382BDBM533382(US11220510, Example 19)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533385BDBM533385(US11220510, Example 22)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533384BDBM533384(US11220510, Example 21)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533393BDBM533393(US11220510, Example 24)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533387BDBM533387(US11220510, Example 23)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533395BDBM533395(US11220510, Example 26)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533394BDBM533394(US11220510, Example 25)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533398BDBM533398(US11220510, Example 28)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533397BDBM533397(US11220510, Example 27)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533400BDBM533400(US11220510, Example 30 | US20250041310, Compound 2...)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533399BDBM533399(US11220510, Example 29)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533344BDBM533344(US11220510, Example 2 | US20250041310, Compound 17)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533359BDBM533359(US11220510, Example 4 | US20250041310, Compound 19)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533358BDBM533358(US11220510, Example 3 | US20250041310, Compound 18)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533361BDBM533361(US11220510, Example 6)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533360BDBM533360(US11220510, Example 5)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533364BDBM533364(US11220510, Example 8)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533363BDBM533363(US11220510, Example 7)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533371BDBM533371(US11220510, Example 10)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533370BDBM533370(US11220510, Example 9)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533374BDBM533374(US11220510, Example 12)
Affinity DataKi: <10nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533381BDBM533381(US11220510, Example 18)
Affinity DataKi:  55nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533373BDBM533373(US11220510, Example 11)
Affinity DataKi:  55nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533375BDBM533375(US11220510, Example 13)
Affinity DataKi:  55nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
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US Patent
LigandChemical structure of BindingDB Monomer ID 533380BDBM533380(US11220510, Example 17)
Affinity DataKi:  550nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533249BDBM533249(US11220510, Example 1)
Affinity DataKi:  550nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533376BDBM533376(US11220510, Example 14)
Affinity DataKi:  550nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533379BDBM533379(US11220510, Example 16)
Affinity DataKi:  550nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Incyte

US Patent
LigandChemical structure of BindingDB Monomer ID 533378BDBM533378(US11220510, Example 15)
Affinity DataKi:  550nMAssay Description:Assays were conducted in black low volume 384-well polystyrene plates (Greiner 784076-25) in a final volume of 10 μL. Test compounds were first ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/14/2022
Entry Details
US Patent