Compile Data Set for Download or QSAR
Report error Found 182 Enz. Inhib. hit(s) with all data for entry = 10558
LigandPNGBDBM550148(3-(5-amino-6-(2-methylthiazol-5- yl)pyrazin-2-yl)-...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550148(3-(5-amino-6-(2-methylthiazol-5- yl)pyrazin-2-yl)-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550149(3-(5-amino-6-(1-(methyl-d3)-1H- 1,2,4-triazol-3-yl...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550149(3-(5-amino-6-(1-(methyl-d3)-1H- 1,2,4-triazol-3-yl...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550150(3-(5-amino-6-(1H-pyrazol-1- yl)pyrazin-2-yl)-N-(1-...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550150(3-(5-amino-6-(1H-pyrazol-1- yl)pyrazin-2-yl)-N-(1-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550151(3-(5-amino-6-(oxazol-5- yl)pyrazin-2-yl)-N-(1- aza...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550152(US11306079, Example 95)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550152(US11306079, Example 95)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549582(US11306079, Example 1)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549582(US11306079, Example 1)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549585(US11306079, Example 65 | 3-(5-Amino-6-(2-methylthi...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549585(US11306079, Example 65 | 3-(5-Amino-6-(2-methylthi...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549592(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549592(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549796(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549796(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549798(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549798(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549799(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549799(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549908(3-(5-amino-6-(1,3-dimethyl-1H-pyrazol-4- yl)pyrazi...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549910(US11306079, Example 16)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549910(US11306079, Example 16)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549911(US11306079, Example 17)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549916(US11306079, Example 18)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549929(3-(5-Amino-6-(2-cyanopyridin-4- yl)pyrazin-2-yl)-N...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549929(3-(5-Amino-6-(2-cyanopyridin-4- yl)pyrazin-2-yl)-N...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549938(3-(5-Amino-6-(3-fluoropyridin-4- yl)pyrazin-2-yl)-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549960(3-(5-Amino-6-(2- (trifluoromethyl)pyridin-4-yl)pyr...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549874(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549874(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549875(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549875(3-(5-Amino-6-(2-methylthiazol-5-yl)pyrazin-2- yl)-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549878(US11306079, Example 9)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549878(US11306079, Example 9)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549893(US11306079, Example 10)
Affinity DataIC50: 100nMAssay Description:[γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549893(US11306079, Example 10)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549894(3-(5-Amino-6-(1,3-dimethyl-1H-pyrazol-4- yl)pyrazi...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549895(3-(5-Amino-6-(1,3-dimethyl-1H-pyrazol-4- yl)pyrazi...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549896(3-(5-Amino-6-(1,3-dimethyl-1H-pyrazol-4- yl)pyrazi...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM549907(3-(5-Amino-6-(1,3-dimethyl-1H-pyrazol-4- yl)pyrazi...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550092(US11306079, Example 31)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550093(US11306079, Example 32)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550094(3-(3-(5-Amino-6-(1H-1,2,4-triazol-1- yl)pyrazin-2-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550095(3-(5-Amino-6-(1H-1,2,4-triazol-1- yl)pyrazin-2-yl)...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550096(3-(3-(5-Amino-6-(1H-1,2,4-triazol-1- yl)pyrazin-2-...)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550097(US11306079, Example 36)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550098(US11306079, Example 37)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

LigandPNGBDBM550099(US11306079, Example 39)
Affinity DataIC50: 100nMAssay Description:γ-33P]ATP (10 mCi/mL) and Wheat Germ Agglutinin (WGA) YSi SPA Scintillation Beads was purchased from Perkin-Elmer (Waltham, Mass.). Lipid kinase...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2022
Entry Details
US Patent

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