Compile Data Set for Download or QSAR
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Found 41 Enz. Inhib. hit(s) with all data for entry = 10723
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562066(US11401255, Compound # 1)
Affinity DataEC50:  371nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562107(US11401255, Compound # 46)
Affinity DataEC50:  203nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562069(US11401255, Compound # 3)
Affinity DataEC50:  405nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562070(US11401255, Compound # 4)
Affinity DataEC50:  164nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562071(US11401255, Compound # 5)
Affinity DataEC50:  63nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562072(US11401255, Compound # 6)
Affinity DataEC50:  2.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562073(US11401255, Compound # 7)
Affinity DataEC50:  2.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562074(US11401255, Compound # 8)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562075(US11401255, Compound # 9)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562076(US11401255, Compound # 10)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562077(US11401255, Compound # 11)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562078(US11401255, Compound # 12)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562079(US11401255, Compound # 13)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562080(US11401255, Compound # 14)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562081(US11401255, Compound # 15)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562082(US11401255, Compound # 16)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562083(US11401255, Compound # 17)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562084(US11401255, Compound # 18)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562085(US11401255, Compound # 19)
Affinity DataEC50:  1.00E+4nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562086(US11401255, Compound # 20)
Affinity DataEC50:  1.00E+4nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562087(US11401255, Compound # 21)
Affinity DataEC50:  238nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562088(US11401255, Compound # 22)
Affinity DataEC50:  246nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562089(US11401255, Compound # 23)
Affinity DataEC50:  272nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562090(US11401255, Compound # 24)
Affinity DataEC50:  190nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562091(US11401255, Compound # 25)
Affinity DataEC50:  382nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562092(US11401255, Compound # 26)
Affinity DataEC50:  938nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562093(US11401255, Compound # 27)
Affinity DataEC50:  190nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562094(US11401255, Compound # 28)
Affinity DataEC50:  134nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562095(US11401255, Compound # 29)
Affinity DataEC50:  2.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562096(US11401255, Compound # 30)
Affinity DataEC50:  5.00E+3nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562097(US11401255, Compound # 31)
Affinity DataEC50:  990nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562098(US11401255, Compound # 32)
Affinity DataEC50:  36nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562099(US11401255, Compound # 33)
Affinity DataEC50:  111nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562100(US11401255, Compound # 35)
Affinity DataEC50:  1.00E+4nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562101(US11401255, Compound # 36)
Affinity DataEC50: >1.00E+4nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562102(US11401255, Compound # 40)
Affinity DataEC50: >1.00E+4nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562103(US11401255, Compound # 42)
Affinity DataEC50:  707nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562104(US11401255, Compound # 43)
Affinity DataEC50:  280nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562105(US11401255, Compound # 44)
Affinity DataEC50:  438nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562106(US11401255, Compound # 45)
Affinity DataEC50:  366nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetE3 ubiquitin-protein ligase parkin(Human)
Mayo Foundation For Medical Education And Research

US Patent
LigandPNGBDBM562068(US11401255, Compound # 2)
Affinity DataEC50:  549nMAssay Description:Ub-charging of E2 enzyme was performed for 90 min at 30° C. in a reaction containing 0.1 μM GST-E1, 3.3 μM E2/UbcH7, 10 μM FLAG-Ub and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent