Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 10797
TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570089BDBM570089(US11427591, Compound 121)
Affinity DataIC50: 7.36nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 50543781BDBM50543781(CHEMBL4632409 | US11427591, Compound 1)
Affinity DataIC50: 9.72nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570092BDBM570092(US11427591, Compound 112)
Affinity DataIC50: 11.5nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570093BDBM570093(US11427591, Compound 113)
Affinity DataIC50: 12.1nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570099BDBM570099(US11427591, Compound 118)
Affinity DataIC50: 13.7nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570094BDBM570094(US11427591, Compound 114)
Affinity DataIC50: 14nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570086BDBM570086(US11427591, Compound 120)
Affinity DataIC50: 14.6nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570084BDBM570084(US11427591, Compound 110)
Affinity DataIC50: 17.3nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570096BDBM570096(US11427591, Compound 115)
Affinity DataIC50: 19.3nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570090BDBM570090(US11427591, Compound 111)
Affinity DataIC50: 24.5nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570097BDBM570097(US11427591, Compound 116)
Affinity DataIC50: 25.8nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570098BDBM570098(US11427591, Compound 117)
Affinity DataIC50: 29.1nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Insilico Medicine Ip

US Patent
LigandChemical structure of BindingDB Monomer ID 570085BDBM570085(US11427591, Compound 119)
Affinity DataIC50: 106nMAssay Description:The activity of the inhibitor compounds against DDR1 and DDR2 was tested using KinaseProfiler (Eurofins). Human DDR1/DDR2 kinase was incubated with 8...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2022
Entry Details
US Patent