Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 10819
TargetAdenosine receptor A2a(Rat)
Inxmed (Nanjing)

US Patent
LigandPNGBDBM571388(US11440916, HZ10136)
Affinity DataIC50: 1.10nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Rat)
Inxmed (Nanjing)

US Patent
LigandPNGBDBM50202993(2-furan-2-yl-7-[2-(4-phenyl-piperazin-1-yl)-ethyl]...)
Affinity DataIC50: 1.20nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Rat)
Inxmed (Nanjing)

US Patent
LigandPNGBDBM50048466(CHEMBL17127 | SCH58261 | 2-(furan-2-yl)-7-phenethy...)
Affinity DataIC50: 1.80nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Rat)
Inxmed (Nanjing)

US Patent
LigandPNGBDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataIC50: 2.5nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Rat)
Inxmed (Nanjing)

US Patent
LigandPNGBDBM86760(CAS_104924 | NSC_104924 | CGS 21680 | US11440916, ...)
Affinity DataIC50: 66.9nMAssay Description:The IC50 (nM) values of the example compound HZ10126 and several reference compounds against the rat A2A receptor were measured in an in vitro assay,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent