Compile Data Set for Download or QSAR
maximum 50k data
Found 49 Enz. Inhib. hit(s) with all data for entry = 10869
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575763(US11465984, Example P42)
Affinity DataIC50:  2.70nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575747(2-(2-chlorophenyl)- 1-(7-fluoro-5- (2-((1-methyl-1...)
Affinity DataIC50:  3nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575740(2-(2-chloropyridin-3-yl)-1-(7-fluoro-5-(2-((1-meth...)
Affinity DataIC50:  3.30nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575778(2-(2-chloropyridin- 3-yl)-1-(7-fluoro-3- methyl-5-...)
Affinity DataIC50:  4.80nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575736(2-(2-chloropyridin- 3-yl)-1-(7- fluoro-5-(2- ((tet...)
Affinity DataIC50:  8.20nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575779(US11465984, Example P60)
Affinity DataIC50:  10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575769(2-(2-chloropyridin- 3-yl)-1-(7-fluoro- 2-methyl-5-...)
Affinity DataIC50: <10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575741(2-(2- chloropyridin- 3-yl)-1-(7- fluoro-5-(2- ((1-...)
Affinity DataIC50: <10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575770(2-(2-chloropyridin- 3-yl)-1-(7-fluoro-2- (methoxym...)
Affinity DataIC50: <10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575752(2-(2-chlorophenyl)- 1-(7-fluoro-5- (2-((1-methyl-1...)
Affinity DataIC50: <10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575753(2-(2- chloropyridin-3- yl)-1-(7-fluoro- 2-methyl-5...)
Affinity DataIC50: <10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575766(1-(7-fluoro-5-(2- ((1-methyl-1H- pyrazol-5-yl) ami...)
Affinity DataIC50: <10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575777(2-(2-chloropyridin- 3-yl)-1-(7-fluoro-2- (methoxym...)
Affinity DataIC50: <10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575768(2-(2-chloropyridin- 3-yl)-1-(7-fluoro-5- (5-methyl...)
Affinity DataIC50: <10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575740(2-(2-chloropyridin-3-yl)-1-(7-fluoro-5-(2-((1-meth...)
Affinity DataIC50: <10nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575757(2-(2-chloro-4- fluorophenyl)-1- (7-fluoro-5-(2- ((...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575758(2-(3-chloropyridin- 4-yl)-1-(7-fluoro- 5-(2-((1-me...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575759(2-(2-chloro-5- fluorophenyl)-1- (7-fluoro-5-(2-((1...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575761(US11465984, Example P40)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575762(US11465984, Example P41)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575764(US11465984, Example P43)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575765(2-(2-chloropyridin- 3-yl)-1-(7-fluoro-5- (6-((1-me...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575756(US11465984, Example P35)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575755(2-(5-chloro-2- fluorophenyl)- 1-(7-fluoro-5- (2-((...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575754(2-(2-chloro-4- fluoropyridin-3-yl)- 1-(7-fluoro-5-...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575751(2-(2-(7-fluoro-5- (2-((1-methyl-1H- pyrazol-5-yl) ...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575750(2-(6-chloropyridin- 2-yl)-1-(7-fluoro- 5-(2-((1-me...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575749(2-(3-chloropyridin- 2-yl)-1-(7-fluoro- 5-(2-((1-me...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575746(1-(7-fluoro-5-(2-((1-methyl-1H-pyrazol-5-yl)amino)...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575745(1-(7-chloro-5- (2-((1-methyl- 1H-pyrazol- 5-yl)ami...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575743(2-(2,4- difluorophenyl)- 1-(7-fluoro-5- (2-((1-met...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575742(1-(7-chloro-5- (2-((1-methyl- 1H-pyrazol- 5-yl)ami...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575738(2-(2-chloropyridin- 3-yl)-1-(7- fluoro-5-(2-((4- h...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575737(2-(2-chloropyridin- 3-yl)-1-(7- fluoro-5-(2- ((tet...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575735(2-(2-chloropyridin- 3-yl)-1-(7- fluoro-5-(2-((3- h...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575734(2-(2-chloropyridin- 3-yl)-1-(7- fluoro-5-(2-((4- h...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575780(2-(2-chloropyridin- 3-yl)-1-(5-(2- (cyclopropylami...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575733(2-(2-chloropyridin- 3-yl)-1-(7- fluoro-5-(2-((2- h...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575775(2-(4-chloropyridin- 3-yl)-1-(7-fluoro- 5-(2-((1-me...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575774(3-(2-chloropyridin- 3-yl)-1-(7-fluoro- 5-(2-((1-me...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575773(2-(2-chloro-3- fluorophenyl)-1- (7-fluoro-5-(2-((1...)
Affinity DataIC50:  55nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575744(2-(2- chloropyridin-3- yl)-1-(7-methyl- 5-(2-((1-m...)
Affinity DataIC50:  550nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575739(2-(2-chloropyridin-3-yl)-1-(7-fluoro-5-(2-((1-hydr...)
Affinity DataIC50:  550nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575732(2-(2-chloropyridin-3-yl)-1-(7-fluoro-5-(2-((1-hydr...)
Affinity DataIC50:  550nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575776(1-(7-fluoro-5-(2- ((1-methyl-1H- pyrazol-5-yl) ami...)
Affinity DataIC50:  550nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575772(2-(2- chloropyridin-3- yl)-1-(7-fluoro- 5-(2-((3- ...)
Affinity DataIC50:  550nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575771(2-(2-chloropyridin- 3-yl)-1-(4,7- difluoro-5-(2-((...)
Affinity DataIC50:  550nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575748(2-(4-chlorophenyl)- 1-(7-fluoro-5- (2-((1-methyl-1...)
Affinity DataIC50:  550nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Shanghai Haihe Pharmaceutical

US Patent
LigandPNGBDBM575760(2-(2,5- difluorophenyl)- 1-(7-fluoro-5- (2-((1-met...)
Affinity DataIC50:  550nMAssay Description:The substrate Z′-LYTE™ Ser/Thr 3 Peptide, the phosphorylation substrate Z′-LYTE™ Ser/Thr 3 Phospho-peptide, 1× kinase buffer (5× kinase b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent