Compile Data Set for Download or QSAR
Report error Found 197 Enz. Inhib. hit(s) with all data for entry = 10907
TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577220BDBM577220(US11472811, Example 18B)
Affinity DataIC50: 0.400nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577340BDBM577340(US11472811, Example 111B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 0.5nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577339BDBM577339(US11472811, Example 111 | 2-(5-amino-2-(furan-2-yl...)
Affinity DataIC50: 0.600nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577217BDBM577217(US11472811, Example 17B)
Affinity DataIC50: 0.600nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577336BDBM577336(US11472811, Example 109B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 0.700nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577196BDBM577196(US11472811, Example 1B)
Affinity DataIC50: 0.700nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577204BDBM577204(US11472811, Example 6 | 2-(5-amino-2-(furan-2-yl)-...)
Affinity DataIC50: 0.900nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577218BDBM577218(US11472811, Example 18)
Affinity DataIC50: 0.900nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577343BDBM577343(US11472811, Example 113B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 0.900nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577368BDBM577368(US11472811, Example 142B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 1nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577335BDBM577335(US11472811, Example 109 | 2-(5-amino-2-(furan-2-yl...)
Affinity DataIC50: 1nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577367BDBM577367(US11472811, Example 141B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 1.10nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577235BDBM577235(US11472811, Example 31B)
Affinity DataKi:  1.20nMAssay Description:Binding affinity of test compounds to four human adenosine receptors, A1, A2A, A2B and A3 was determined in radioligand competitive binding assay (co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577366BDBM577366(US11472811, Example 140 | 2-(5-amino-2-(furan-2-yl...)
Affinity DataIC50: 1.20nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577342BDBM577342(US11472811, Example 112B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 1.20nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577269BDBM577269(US11472811, Example 58B)
Affinity DataIC50: 1.30nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 50202986BDBM50202986(SCH-420814 | 7-(2-(4-(2,4-difluorophenyl)piperazin...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity of test compounds to four human adenosine receptors, A1, A2A, A2B and A3 was determined in radioligand competitive binding assay (co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577231BDBM577231(US11472811, Example 29 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 1.30nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577224BDBM577224(US11472811, Example 22 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 1.40nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577194BDBM577194(US11472811, Example 1)
Affinity DataIC50: 1.40nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577205BDBM577205(US11472811, Example 7 | 2-(5-amino-2-(furan-2-yl)-...)
Affinity DataIC50: 1.5nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577227BDBM577227(US11472811, Example 25 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 1.5nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577256BDBM577256(US11472811, Example 48B)
Affinity DataIC50: 1.60nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577292BDBM577292(US11472811, Example 76B)
Affinity DataKi:  1.60nMAssay Description:Binding affinity of test compounds to four human adenosine receptors, A1, A2A, A2B and A3 was determined in radioligand competitive binding assay (co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577283BDBM577283(US11472811, Example 69B)
Affinity DataKi:  1.60nMAssay Description:Binding affinity of test compounds to four human adenosine receptors, A1, A2A, A2B and A3 was determined in radioligand competitive binding assay (co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577230BDBM577230(US11472811, Example 28 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 1.60nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577284BDBM577284(US11472811, Example 70 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 1.70nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577300BDBM577300(US11472811, Example 82B)
Affinity DataKi:  1.70nMAssay Description:Binding affinity of test compounds to four human adenosine receptors, A1, A2A, A2B and A3 was determined in radioligand competitive binding assay (co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577377BDBM577377(US11472811, Example 149B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 1.70nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577267BDBM577267(US11472811, Example 58 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 1.80nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577365BDBM577365(US11472811, Example 139 | 2-(5-amino-2-(furan-2-yl...)
Affinity DataIC50: 1.90nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577346BDBM577346(US11472811, Example 115 | 2-(5-amino-2-(furan-2-yl...)
Affinity DataIC50: 1.90nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577225BDBM577225(US11472811, Example 23 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 1.90nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577379BDBM577379(US11472811, Example 151B | (cis)-4-((R)-2-(5-amino...)
Affinity DataIC50: 2nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577206BDBM577206(US11472811, Example 8 | 2-(5-amino-2-(furan-2-yl)-...)
Affinity DataIC50: 2nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577354BDBM577354(US11472811, Example 119B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 2nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577370BDBM577370(US11472811, Example 144B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 2.10nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577348BDBM577348(US11472811, Example 116 | 2-(5-amino-2-(furan-2-yl...)
Affinity DataIC50: 2.20nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577202BDBM577202(US11472811, Example 4B)
Affinity DataIC50: 2.20nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577256BDBM577256(US11472811, Example 48B)
Affinity DataKi:  2.20nMAssay Description:Binding affinity of test compounds to four human adenosine receptors, A1, A2A, A2B and A3 was determined in radioligand competitive binding assay (co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577292BDBM577292(US11472811, Example 76B)
Affinity DataIC50: 2.20nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577235BDBM577235(US11472811, Example 31B)
Affinity DataIC50: 2.30nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577239BDBM577239(US11472811, Example 33B | (R)-2-(5-amino-2-(furan-...)
Affinity DataIC50: 2.30nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577337BDBM577337(US11472811, Example 110 | 2-(5-amino-2-(furan-2-yl...)
Affinity DataIC50: 2.40nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577278BDBM577278(US11472811, Example 66B | (R)-2-(5-amino-2-(furan-...)
Affinity DataIC50: 2.40nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577334BDBM577334(US11472811, Example 108B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 2.5nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577228BDBM577228(US11472811, Example 26 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 2.60nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577259BDBM577259(US11472811, Example 51 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 2.70nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577254BDBM577254(US11472811, Example 48 | 2-(5-amino-2-(furan-2-yl)...)
Affinity DataIC50: 2.90nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

TargetAdenosine deaminase(Human)
Beigene

US Patent
LigandChemical structure of BindingDB Monomer ID 577338BDBM577338(US11472811, Example 110B | (R)-2-(5-amino-2-(furan...)
Affinity DataIC50: 2.90nMAssay Description:HEK293-A2AR-luc2p/CRE/Hygro cells were seeded at a density of 5,000 cells/well in DMEM with 1% FBS and 1 U/mL adenosine deaminase (ADA) (Sigma). Afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2022
Entry Details
US Patent

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