Compile Data Set for Download or QSAR
Report error Found 143 Enz. Inhib. hit(s) with all data for entry = 10936
TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579718BDBM579718(US11485711, Compound 146 | 3-ethyl-4-((5-(4-iodoph...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579738BDBM579738(US11485711, Compound 180 | N-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579704BDBM579704(US11485711, Compound 109 | N-(4-((5-(4-(1H-imidazo...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579709BDBM579709(US11485711, Compound 119 | 4-((5-(5-chlorothiophen...)
Affinity DataIC50: 1nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579739BDBM579739(US11485711, Compound 181 | N-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 2nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579693BDBM579693(US11485711, Compound 81 | 3-ethyl-4-((5-(4- hydrox...)
Affinity DataKd:  3nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579743BDBM579743(US11485711, Compound 187 | N-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 3nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579689BDBM579689(US11485711, Compound 58 | N-(4-((5-(4-hydroxypheny...)
Affinity DataIC50: 3nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579794BDBM579794(US11485711, Compound 265 | 4-((5-(4-(1H-pyrazol-4-...)
Affinity DataIC50: 4nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579686BDBM579686(US11485711, Compound 39 | 4-((5-(4-hydroxyphenyl)-...)
Affinity DataKd:  6nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579714BDBM579714(US11485711, Compound 140 | 4-((5-(1H-indol-3-yl)-1...)
Affinity DataIC50: 6nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579761BDBM579761(US11485711, Compound 205 | 1-(4-(3-((4-hydroxy-2- ...)
Affinity DataIC50: 6nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579764BDBM579764(US11485711, Compound 208 | methyl (4-((5-(4-(1H-py...)
Affinity DataIC50: 7nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579740BDBM579740(US11485711, Compound 182 | 2-(dimethylamino)-N-(4-...)
Affinity DataIC50: 7nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579799BDBM579799(US11485711, Compound 276 | 3-methyl-4-((5-(4-(1-me...)
Affinity DataIC50: 8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579736BDBM579736(US11485711, Compound 176 | 4-((5-(4-(1H-imidazol-1...)
Affinity DataIC50: 8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579705BDBM579705(US11485711, Compound 110 | N-(4-((5-(4-(1H-imidazo...)
Affinity DataIC50: 8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579691BDBM579691(US11485711, Compound 62 | 4-((4-fluoro-5-(4- hydro...)
Affinity DataKd:  8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579763BDBM579763(US11485711, Compound 207 | 1-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 8nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579687BDBM579687(US11485711, Compound 40 | 4-((5-(4-hydroxyphenyl)-...)
Affinity DataKd:  9nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579765BDBM579765(US11485711, Compound 209 | ethyl (4-((5-(4-(1H-pyr...)
Affinity DataIC50: 9nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579801BDBM579801(US11485711, Compound 278 | 3-methyl-4-((5-(4-(3- (...)
Affinity DataIC50: 9nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579708BDBM579708(US11485711, Compound 117 | 4-((5-(benzo[b]thiophen...)
Affinity DataIC50: 10nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579741BDBM579741(US11485711, Compound 183 | N-(4-((5-(3-fluoro-4- h...)
Affinity DataIC50: 10nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579689BDBM579689(US11485711, Compound 58 | N-(4-((5-(4-hydroxypheny...)
Affinity DataKd:  11nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579800BDBM579800(US11485711, Compound 277 | 4-((5-(4-(3,5-dimethyl-...)
Affinity DataIC50: 11nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579703BDBM579703(US11485711, Compound 86 | N-(4-((5-(4-hydroxy-3- m...)
Affinity DataIC50: 12nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579693BDBM579693(US11485711, Compound 81 | 3-ethyl-4-((5-(4- hydrox...)
Affinity DataIC50: 12nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579696BDBM579696(US11485711, Compound 94 | 2-fluoro-4-((5-(4- hydro...)
Affinity DataKd:  12nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579692BDBM579692(US11485711, Compound 73 | 4-((5-(4-(1H-imidazol-1-...)
Affinity DataKd:  14nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579683BDBM579683(US11485711, Compound 24 | 4-((5-(4-aminophenyl)-1H...)
Affinity DataKd:  14nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579735BDBM579735(US11485711, Compound 175 | 4-((5-(4-(1H-inidazol-1...)
Affinity DataIC50: 15nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579730BDBM579730(US11485711, Compound 170 | N-(4-((5-(4-(1H-imidazo...)
Affinity DataIC50: 15nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579690BDBM579690(US11485711, Compound 59 | N-(4-((5-(4-hydroxypheny...)
Affinity DataKd:  16nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579694BDBM579694(US11485711, Compound 88 | 2-fluoro-4-(3-((4-hydrox...)
Affinity DataKd:  16nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579731BDBM579731(US11485711, Compound 171 | N-(4-((5-(4-(1H-imidazo...)
Affinity DataIC50: 16nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579710BDBM579710(US11485711, Compound 126 | 3-chloro-4-((5-(4- hydr...)
Affinity DataIC50: 17nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579688BDBM579688(US11485711, Compound 49 | 3-fluoro-4-((5-(4- hydro...)
Affinity DataKd:  19nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579798BDBM579798(US11485711, Compound 275 | 2-fluoro-4-((5-(4-hydro...)
Affinity DataIC50: 19nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579797BDBM579797(US11485711, Compound 274 | 4-((5-(4-(1H-pyrazol-1-...)
Affinity DataIC50: 20nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579697BDBM579697(US11485711, Compound 111 | 4-((5-(4-(1H-imidazol-1...)
Affinity DataKd:  20nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579695BDBM579695(US11485711, Compound 89 | 4-((5-(4-hydroxyphenyl)-...)
Affinity DataKd:  21nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579713BDBM579713(US11485711, Compound 139 | N-(4-((5-(4-(1H-pyrazol...)
Affinity DataIC50: 22nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579702BDBM579702(US11485711, Compound 85 | 4-(3-((4-hydroxy-2- meth...)
Affinity DataIC50: 23nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579726BDBM579726(US11485711, Compound 158 | N-(4-((5-(3-fluoro-4- h...)
Affinity DataIC50: 23nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579712BDBM579712(US11485711, Compound 138 | 4-((5-(4-(1H-pyrazol-1-...)
Affinity DataIC50: 23nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579770BDBM579770(US11485711, Compound 215 | 1-(4-(3-((4-hydroxy-2- ...)
Affinity DataIC50: 24nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579804BDBM579804(US11485711, Compound 281 | methyl (4-((5-(4-(1H-py...)
Affinity DataIC50: 25nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579684BDBM579684(US11485711, Compound 29 | N1-(5-(4-chlorophenyl)-1...)
Affinity DataKd:  25nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

TargetTRAF2 and NCK-interacting protein kinase(Human)
Korea Research Institute of Chemical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 579727BDBM579727(US11485711, Compound 160 | 4-(3-((2-ethyl-4- hydro...)
Affinity DataIC50: 26nMAssay Description:The inhibitory properties of compounds were evaluated with TNIK kinase enzyme system and luminescent ADP-GloFigure US11485711-20221101-P00001 Kinase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2023
Entry Details
US Patent

Displayed 1 to 50 (of 143 total ) | Next | Last >>
Jump to: