Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 10976
TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581757BDBM581757(US11512087, Example 1)
Affinity DataIC50: 2.10nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581831BDBM581831(US11512087, Example 13-1)
Affinity DataIC50: 3.30nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581837BDBM581837(US11512087, Example 25)
Affinity DataIC50: 3.40nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581838BDBM581838(US11512087, Example 26-1)
Affinity DataIC50: 3.70nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581832BDBM581832(US11512087, Example 13-9)
Affinity DataIC50: 4.10nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581795BDBM581795(US11512087, Example 4-1)
Affinity DataIC50: 5.10nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581830BDBM581830(US11512087, Example 12)
Affinity DataIC50: 5.10nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581780BDBM581780(US11512087, Example 2)
Affinity DataIC50: 5.40nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581829BDBM581829(US11512087, Example 10)
Affinity DataIC50: 6.90nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581828BDBM581828(US11512087, Example 8)
Affinity DataIC50: 7.60nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581835BDBM581835(US11512087, Example 18-1)
Affinity DataIC50: 7.70nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581806BDBM581806(US11512087, Example 4-3)
Affinity DataIC50: 8.5nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581805BDBM581805(US11512087, Example 4-2)
Affinity DataIC50: 9.30nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581836BDBM581836(US11512087, Example 23)
Affinity DataIC50: 9.70nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581833BDBM581833(US11512087, Example 14-4)
Affinity DataIC50: 12nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581834BDBM581834(US11512087, Example 14-11)
Affinity DataIC50: 50nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetTyrosine-protein kinase Lck(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581806BDBM581806(US11512087, Example 4-3)
Affinity DataIC50: 2.50E+3nMAssay Description:Tyrosine phosphorylation of Lck was performed by using Z′-LYTE Kinase Assay Kit-Tyr 2 Peptide (Invitrogen) containing the following reagents (T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetTyrosine-protein kinase Lck(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581831BDBM581831(US11512087, Example 13-1)
Affinity DataIC50: 1.00E+4nMAssay Description:Tyrosine phosphorylation of Lck was performed by using Z′-LYTE Kinase Assay Kit-Tyr 2 Peptide (Invitrogen) containing the following reagents (T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent

TargetTyrosine-protein kinase Lck(Human)
Ono Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 581757BDBM581757(US11512087, Example 1)
Affinity DataIC50: 1.00E+4nMAssay Description:Tyrosine phosphorylation of Lck was performed by using Z′-LYTE Kinase Assay Kit-Tyr 2 Peptide (Invitrogen) containing the following reagents (T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2023
Entry Details
US Patent