Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 10995
TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582503BDBM582503(US11524941, Compound 10)
Affinity DataIC50: 97.9nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582508BDBM582508(US11524941, Compound 22)
Affinity DataIC50: 112nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582514BDBM582514(US11524941, Compound 35)
Affinity DataIC50: 186nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582506BDBM582506(US11524941, Compound 18)
Affinity DataIC50: 194nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582502BDBM582502(US11524941, Compound 9)
Affinity DataIC50: 228nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582505BDBM582505(US11524941, Compound 15)
Affinity DataIC50: 275nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582511BDBM582511(US11524941, Compound 31)
Affinity DataIC50: 290nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582513BDBM582513(US11524941, Compound 34)
Affinity DataIC50: 303nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582515BDBM582515(US11524941, Compound 36)
Affinity DataIC50: 308nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582510BDBM582510(US11524941, Compound 29)
Affinity DataIC50: 308nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582500BDBM582500(US11524941, Compound 1)
Affinity DataIC50: 330nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582507BDBM582507(US11524941, Compound 19)
Affinity DataIC50: 349nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582512BDBM582512(US11524941, Compound 32)
Affinity DataIC50: 433nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582509BDBM582509(US11524941, Compound 27)
Affinity DataIC50: 526nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Medshine Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 582504BDBM582504(US11524941, Compound 12)
Affinity DataIC50: 569nMAssay Description:The purpose of this assay was to detect the inhibitory activity of the compounds against LSD1 in vitro. The enzyme used in this assay was human LSD1 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2023
Entry Details
US Patent