Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 11014
TargetAmine oxidase [copper-containing] 2(Human)
Proximagen

US Patent
LigandPNGBDBM585361(4-{4-[3-(4-Chlorophenyl)-3H-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 50nMAssay Description:Briefly, test compounds were dissolved in dimethyl sulfoxide (DMSO) to a concentration of 10 mM. Dose-response measurements were assayed by either cr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 2(Human)
Proximagen

US Patent
LigandPNGBDBM585359(1-({5-[3-(4-Fluorophenyl)-3H- imidazo[4,5-c]pyridi...)
Affinity DataIC50: 50nMAssay Description:Briefly, test compounds were dissolved in dimethyl sulfoxide (DMSO) to a concentration of 10 mM. Dose-response measurements were assayed by either cr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 2(Human)
Proximagen

US Patent
LigandPNGBDBM585360(2-Methyl-1-({5-[3-(4- methylphenyl)-3H- imidazo[...)
Affinity DataIC50: 50nMAssay Description:Briefly, test compounds were dissolved in dimethyl sulfoxide (DMSO) to a concentration of 10 mM. Dose-response measurements were assayed by either cr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 2(Human)
Proximagen

US Patent
LigandPNGBDBM585357(5-[3-(4-Fluorophenyl)-3H-imidazo[4,5-c]pyridin-2-y...)
Affinity DataIC50: 125nMAssay Description:Briefly, test compounds were dissolved in dimethyl sulfoxide (DMSO) to a concentration of 10 mM. Dose-response measurements were assayed by either cr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 2(Human)
Proximagen

US Patent
LigandPNGBDBM585358(5-[3-(4-Fluorophenyl)-3H- imidazo[4,5-c]pyridin-2-...)
Affinity DataIC50: 350nMAssay Description:Briefly, test compounds were dissolved in dimethyl sulfoxide (DMSO) to a concentration of 10 mM. Dose-response measurements were assayed by either cr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 2(Human)
Proximagen

US Patent
LigandPNGBDBM585362(6-{4-[3-(4-Chlorophenyl)-3H-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 350nMAssay Description:Briefly, test compounds were dissolved in dimethyl sulfoxide (DMSO) to a concentration of 10 mM. Dose-response measurements were assayed by either cr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 2(Human)
Proximagen

US Patent
LigandPNGBDBM585365(3-(4-Fluorophenyl)-N-(oxan-4-ylmethyl)-3H-imidazo[...)
Affinity DataIC50: 350nMAssay Description:Briefly, test compounds were dissolved in dimethyl sulfoxide (DMSO) to a concentration of 10 mM. Dose-response measurements were assayed by either cr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 2(Human)
Proximagen

US Patent
LigandPNGBDBM585363(3-{[3-(4-Chlorophenyl)-3H-imidazo[4,5-c]pyridin-2-...)
Affinity DataIC50: 350nMAssay Description:Briefly, test compounds were dissolved in dimethyl sulfoxide (DMSO) to a concentration of 10 mM. Dose-response measurements were assayed by either cr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

TargetAmine oxidase [copper-containing] 2(Human)
Proximagen

US Patent
LigandPNGBDBM585364(1-{3-[3-(4-chlorophenyl)-3H-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 350nMAssay Description:Briefly, test compounds were dissolved in dimethyl sulfoxide (DMSO) to a concentration of 10 mM. Dose-response measurements were assayed by either cr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

LigandPNGBDBM585361(4-{4-[3-(4-Chlorophenyl)-3H-imidazo[4,5-c]pyridin-...)
Affinity DataIC50: 505nMAssay Description:Compounds of the invention were tested for inhibition of the human ether a go-go related gene (hERG) K+ channel using IonWorks patch clamp electrophy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent

LigandPNGBDBM585359(1-({5-[3-(4-Fluorophenyl)-3H- imidazo[4,5-c]pyridi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Compounds of the invention were tested for inhibition of the human ether a go-go related gene (hERG) K+ channel using IonWorks patch clamp electrophy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2023
Entry Details
US Patent