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Found 46 Enz. Inhib. hit(s) with all data for entry = 11076
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466133(CHEMBL4292847 | US11547712, Compound 3-1)
Affinity DataKd:  7.30E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582867(US11547712, Compound 14-7)
Affinity DataKd:  1.20E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582657(US11547712, Compound 3-8)
Affinity DataKd:  3.40E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582658(US11547712, Compound 3-9)
Affinity DataKd:  3.10E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582659(US11547712, Compound 3-10)
Affinity DataKd:  650nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582660(US11547712, Compound 3-11)
Affinity DataKd:  1.10E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466136(CHEMBL4292463 | US11547712, Compound 3-12)
Affinity DataKd:  185nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466135(CHEMBL4284570 | US11547712, Compound 3-13)
Affinity DataKd:  420nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466148(CHEMBL4288534 | US11547712, Compound 3-14)
Affinity DataKd:  840nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466137(CHEMBL4280328 | US11547712, Compound 3-15)
Affinity DataKd:  71nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466153(CHEMBL4293751 | US11547712, Compound 3-16)
Affinity DataKd:  900nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466138(CHEMBL4283169 | US11547712, Compound 3-17)
Affinity DataKd:  810nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466152(CHEMBL4285515 | US11547712, Compound 3-18)
Affinity DataKd:  1.30E+4nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466139(CHEMBL4284175 | US11547712, Compound 3-19)
Affinity DataKd:  660nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466131(CHEMBL4282090 | US11547712, Compound 3-20)
Affinity DataKd:  7.70E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466149(CHEMBL4289970 | US11547712, Compound 3-21)
Affinity DataKd:  6.20E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466140(CHEMBL4283581 | US11547712, Compound 3-22)
Affinity DataKd:  320nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466134(CHEMBL4291431 | US11547712, Compound 3-23)
Affinity DataKd:  860nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466154(CHEMBL4277463 | US11547712, Compound 3-24)
Affinity DataKd:  2.20E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582707(US11547712, Compound 4-1)
Affinity DataKd:  460nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466141(CHEMBL4288107 | US11547712, Compound 4-2)
Affinity DataKd:  440nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466142(CHEMBL4280876 | US11547712, Compound 3-25)
Affinity DataKd:  1.10E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466155(CHEMBL4291519 | US11547712, Compound 3-26)
Affinity DataKd:  2.30E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582722(US11547712, Compound 3-27)
Affinity DataKd:  3.00E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466143(CHEMBL4284277 | US11547712, Compound 3-28)
Affinity DataKd:  1.90E+4nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466132(CHEMBL4294914 | US11547712, Compound 3-29)
Affinity DataKd:  7.00E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466144(CHEMBL4289634 | US11547712, Compound 3-30)
Affinity DataKd:  1.40E+4nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466151(CHEMBL4276858 | US11547712, Compound 3-31)
Affinity DataKd:  3.80E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582850(US11547712, Compound 3-32)
Affinity DataKd:  1.60E+4nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582851(US11547712, Compound 3-33)
Affinity DataKd:  7.80E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466145(CHEMBL4282379 | US11547712, Compound 3-34)
Affinity DataKd:  1.60E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582853(US11547712, Compound 3-35)
Affinity DataKd:  1.50E+4nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582854(US11547712, Compound 3-36)
Affinity DataKd:  1.70E+4nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466156(CHEMBL4290892 | US11547712, Compound 3-37)
Affinity DataKd:  950nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466150(CHEMBL4277245 | US11547712, Compound 3-38)
Affinity DataKd:  1.60E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466146(CHEMBL4285200 | US11547712, Compound 3-39)
Affinity DataKd:  2.20E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466147(CHEMBL4288550 | US11547712, Compound 3-41)
Affinity DataKd:  7.30E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582859(US11547712, Compound 3-47)
Affinity DataKd:  1.40E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582860(US11547712, Compound 3-48)
Affinity DataKd:  3.70E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582861(US11547712, Compound 3-49)
Affinity DataKd:  4.30E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582862(US11547712, Compound 14-1)
Affinity DataKd:  4.30E+4nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582863(US11547712, Compound 14-2)
Affinity DataKd:  3.70E+4nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582864(US11547712, Compound 14-3)
Affinity DataKd:  8.80E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582865(US11547712, Compound 14-4)
Affinity DataKd:  1.70E+4nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM582866(US11547712, Compound 14-5)
Affinity DataKd:  6.80E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Icahn School Of Medicine At Mount Sinai

US Patent
LigandPNGBDBM50466133(CHEMBL4292847 | US11547712, Compound 3-1)
Affinity DataKd:  4.50E+3nMAssay Description:Compound 1, a 1,3,4-thiadiazine compound identified in a screening assay, was evaluated for testing of in vitro DYRK1A activity at 30 μM concent...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent