Compile Data Set for Download or QSAR
Report error Found 471 Enz. Inhib. hit(s) with all data for entry = 11184
TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418452BDBM418452(1-(3-Fluoro-5-methylpyridin- 2-yl)-7-methoxy-3-met...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418477BDBM418477(7-Methoxy-3-methyl-1-(3- methyl-1H-pyrazol-4-yl)-8...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418453BDBM418453(1-(1,3-Dimethyl-1H-pyrazol- 4-yl)-8-(1-ethyl-1H-py...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418448BDBM418448(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoropyrid...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418472BDBM418472(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoro-5-methylp...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418473BDBM418473(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoro-5-me...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418465BDBM418465(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoropyridin-4-...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418473BDBM418473(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoro-5-me...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418472BDBM418472(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoro-5-methylp...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418477BDBM418477(7-Methoxy-3-methyl-1-(3- methyl-1H-pyrazol-4-yl)-8...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418450BDBM418450(1-(3-Fluoro-5-methylpyridin- 4-yl)-7-methoxy-3-met...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418435BDBM418435(1-[5-(azetidin-3-ylmethoxy)-3-fluoropyridin-2-yl]-...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418515BDBM418515(1-(3-Fluoro-5-fluoro- methoxypyridin-2-yl)-7- meth...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418513BDBM418513(1-(3,5-Difluoropyridin-2-yl)- 8-(1,3-dimethyl-1H-p...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418519BDBM418519(1-(5-Difluoromethoxy-3- fluoropyridin-2-yl)-7- met...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418457BDBM418457(1-(3-Ethyl-5-fluoropyridin-4- yl)-8-(1-ethyl-1H-py...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418518BDBM418518(1-(5-Ethoxy-3-fluoropyridin- 2-yl)-7-methoxy-3-met...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418458BDBM418458(1-(3,5-Difluoropyridin-4-yl)- 8-(1-ethyl-1H-pyrazo...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418524BDBM418524(1-(5-Chloro-3-fluoropyridin- 2-yl)-7-methoxy-3-met...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418436BDBM418436(US10457677, Example 4 | US10745399, Example 4 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418437BDBM418437(US10457677, Example 5 | US10745399, Example 5 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418527BDBM418527(1-(3-Fluoro-5-methoxy- pyridin-2-yl)-7-methoxy-3- ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418525BDBM418525(7-Methoxy-3-methyl-8-(1- methyl-1H-pyrazol-4-yl)-1...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418503BDBM418503(1-[3-Fluoro-5-(2-hydroxy- ethoxy)-2-pyridyl]-7- me...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418502BDBM418502(1-[3-Fluoro-5-(2-methoxy- ethoxy)-2-pyridyl]-7- me...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418454BDBM418454(1-(3,5-Difluoropyridin-4-yl)- 7-methoxy-3-methyl-8...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418501BDBM418501(8-(3-Amino-1H-pyrazol-5- yl)-1-(3-fluoro-2-pyridyl...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418505BDBM418505(7-Methoxy-3-methyl-8-(1- methyl-1H-pyrazol-4-yl)-1...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418456BDBM418456(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoropyridin-2-...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418512BDBM418512(1-(3,5-Difluoropyridin-2-yl)- 7-methoxy-8-(1-methy...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418511BDBM418511(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoro-5- m...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418510BDBM418510(1-(3-Fluoro-5-methoxy- pyridin-2-yl)-7-methoxy-3- ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418434BDBM418434(US10457677, Example 2 | US10745399, Example 2 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418548BDBM418548(8-(1-Difluoromethyl-1H- pyrazol-4-yl)-1-(3-fluoro-...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418547BDBM418547(8-(1-Ethyl-3-methyl-1H- pyrazol-4-yl)-1-(3-fluoro-...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418440BDBM418440(US10457677, Example 8 | US10745399, Example 8 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418545BDBM418545(1-(3-Fluoro-5-methoxy- pyridin-4-yl)-8-(1-fluoro- ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418552BDBM418552(1-(3-Difluoromethoxy-5- fluoropyridin-4-yl)-8-(1,3...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418441BDBM418441(US10457677, Example 9 | US10745399, Example 9 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418551BDBM418551(1-(3-Difluoromethoxy-5- fluoropyridin-4-yl)-7- met...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 598110BDBM598110(US11608338, Example 145 | 1-[3-Fluoro-5-(trideuter...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418549BDBM418549(1-(3-Fluoro-5-methoxy- pyridin-2-yl)-7-methoxy-3- ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 598115BDBM598115(US11608338, Example 150 | 8-(1,3-Dimethylpyrazol-4...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418554BDBM418554(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoro-5-fl...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418553BDBM418553(1-(3-Fluoro-5-fluoro- methoxypyridin-4-yl)-7- meth...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 598120BDBM598120(US11608338, Example 155 | 1-[3-Fluoro-5-(trideuter...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418559BDBM418559(1-(1,3-Dimethyl-1H-pyrazol- 4-yl)-7-methoxy-3-meth...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418442BDBM418442(US10457677, Example 10 | US10745399, Example 10 | ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418557BDBM418557(1-(3-Fluoro-5-methoxy- pyridin-4-yl)-7-methoxy-3- ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418530BDBM418530(1-(3-Ethyl-5-fluoropyridin-4- yl)-7-methoxy-3-meth...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
US Patent

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