Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 11300
TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605508(US11673884, Compound AC-2)
Affinity DataIC50: 1nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605513(US11673884, Compound AC-6)
Affinity DataIC50: 1nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605512(US11673884, Compound AC-5)
Affinity DataIC50: 1nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605509(US11673884, Compound AC-3)
Affinity DataIC50: 1nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605517(US11673884, Compound AC-10)
Affinity DataIC50: 1nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605516(US11673884, Compound AC-9)
Affinity DataIC50: 1nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605515(US11673884, Compound AC-8)
Affinity DataIC50: 1nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605519(US11673884, Compound AC-12)
Affinity DataIC50: 1nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605518(US11673884, Compound AC-11)
Affinity DataIC50: 1nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605511(US11673884, Compound AC-4)
Affinity DataIC50: 5.5nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605514(US11673884, Compound AC-7)
Affinity DataIC50: 5.5nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent

TargetMacrophage metalloelastase(Human)
Foresee Pharmaceuticals

US Patent
LigandPNGBDBM605455(US11673884, Compound AC-1)
Affinity DataIC50: 55nMAssay Description:The inhibitory effect of compounds on the rate of cleaving fluorogenic MMP substrate (Enzo, BML-P128) by recombinant human MMP-12 catalytic domain (E...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2023
Entry Details
US Patent