Compile Data Set for Download or QSAR
Report error Found 142 Enz. Inhib. hit(s) with all data for entry = 11713
LigandChemical structure of BindingDB Monomer ID 642477BDBM642477(US11851426, Example 103)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642478BDBM642478(US11851426, Example 104)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642479BDBM642479(US11851426, Example 105)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642480BDBM642480(US11851426, Example 106)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642473BDBM642473(N-((3R,4S)-3-Methyl-1- ((1-methyl-1H-pyrazol- 4-yl...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642474BDBM642474(US11851426, Example 100)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642475BDBM642475(US11851426, Example 101)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642476BDBM642476(US11851426, Example 102)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642485BDBM642485(N-((3R,4S)-3-Methyl-1- (methylsulfonyl)piperidin- ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642486BDBM642486(N-((3R,4S)-3-Methyl-1- (methylsulfonyl)piperidin- ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642487BDBM642487(N-((3R,4S)-3-Methyl-1- (methylsulfonyl)piperidin- ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642488BDBM642488(N-((3R,4S)-3-Methyl-1- (methylsulfonyl)piperidin- ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642481BDBM642481(N-((3R,4S)-3-Methyl-1- (methylsulfonyl)piperidin- ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642482BDBM642482(5-(3- (Difluoromethyl) cyclobutoxy)-N- ((3R,4S)-3-...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642483BDBM642483(5-Cyclopropoxy-N- ((3R,4S)-3-methyl-1- (methylsulf...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642484BDBM642484(5-((4,4- Difluorocyclohexyl) oxy)-N-((3R,4S)-3- me...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642461BDBM642461(US11851426, Example 138 | US11851426, Example 139 ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642462BDBM642462(US11851426, Example 88)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642463BDBM642463(US11851426, Example 89)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642464BDBM642464(N-(3R,4S)-3-Methyl-1- (methylsulfonyl)piperidin- 4...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642457BDBM642457(US11851426, Example 83)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642458BDBM642458(N-((3R,4S)-1- (Ethylsulfonyl)-3- methylpiperidin-4...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642459BDBM642459(N-((3R,4S)-1- (Cyclopropylsulfonyl)- 3-methylpiper...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642460BDBM642460(N-((3R,4S)-3-Methyl-1- ((1-methyl-1H- imidazol-4- ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642469BDBM642469(5-Cyclobutoxy-N- ((3R,4S)-3-methyl-1- ((1-methyl-1...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642470BDBM642470(N-((3R,4S)-1- (Ethylsulfonyl)-3- methylpiperidin-4...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642471BDBM642471(N-((3R,4S)-1- (Cyclopropylsulfonyl)- 3-methylpiper...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642472BDBM642472(N-((3R,4S)-3-Methyl-1- (methylsulfonyl)piperidin- ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642465BDBM642465(N-((3R,4S)-1- (Ethylsulfonyl)-3- methylpiperidin-4...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642466BDBM642466(N-((3R,4S)-1- (Cyclopropylsulfonyl)- 3-methylpiper...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642467BDBM642467(5-Cyclobutoxy-N- ((3R,4S)-1- (ethylsulfonyl)-3- me...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642468BDBM642468(5-Cyclobutoxy-N- ((3R,4S)-3-methyl-1- ((1-methyl-1...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642509BDBM642509(US11851426, Example 135)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642510BDBM642510(US11851426, Example 136)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642461BDBM642461(US11851426, Example 138 | US11851426, Example 139 ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642461BDBM642461(US11851426, Example 138 | US11851426, Example 139 ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642505BDBM642505(US11851426, Example 131)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642506BDBM642506(US11851426, Example 132)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642507BDBM642507(US11851426, Example 133)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642508BDBM642508(US11851426, Example 134)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642461BDBM642461(US11851426, Example 138 | US11851426, Example 139 ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642514BDBM642514(5-(Cyclopentyloxy)-N- ((3R,4S)-3-methyl-1- (methyl...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642515BDBM642515(US11851426, Example 142 | 5-Isopropoxy-N-(1- (meth...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642515BDBM642515(US11851426, Example 142 | 5-Isopropoxy-N-(1- (meth...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642493BDBM642493(N-(1- (Methylsulfonyl)piperidin- 4-yl)-6-(1H- pyra...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642494BDBM642494(N-(1- (Methylsulfonyl) piperidin-4-yl)-6-(1H- pyra...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642495BDBM642495(5-(Isopentyloxy)-N-(1- (methylsulfonyl)piperidin- ...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642496BDBM642496(5-Ethoxy-N-(1- (methylsulfonyl)piperidin- 4-yl)-6-...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642489BDBM642489(5- (Cyclopropylmethoxy)- N-((3R,4S)-3-methyl-1- (m...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 642490BDBM642490(5-(Isopentyloxy)-N- ((3R,4S)-3-methyl-1- (methylsu...)
Affinity DataIC50: 20nMAssay Description:CDK2/Cyclin E1 enzyme activity assays utilize full-length human CDK2 co-expressed as N-terminal GST-tagged protein with FLAG-Cyclin E1 in a baculovir...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
US Patent

Displayed 1 to 50 (of 142 total ) | Next | Last >>
Jump to: