Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 12200
TargetSet1/Ash2 histone methyltransferase complex subunit ASH2(Human)
Memorial Sloan-Kettering Cancer Center

US Patent
LigandPNGBDBM685914(US12043645, Example 7)
Affinity DataIC50: 20nMAssay Description:This assay relies on Whatman P-81 filter paper, which binds peptides but not SAM. Protein Methyl Transferases (PMTs) transfer 3H-Me of [3H-Me]-SAM to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2024
Entry Details
US Patent

TargetSet1/Ash2 histone methyltransferase complex subunit ASH2(Human)
Memorial Sloan-Kettering Cancer Center

US Patent
LigandPNGBDBM685904(US12043645, Example 1)
Affinity DataIC50: 390nMAssay Description:This assay relies on Whatman P-81 filter paper, which binds peptides but not SAM. Protein Methyl Transferases (PMTs) transfer 3H-Me of [3H-Me]-SAM to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2024
Entry Details
US Patent

TargetSet1/Ash2 histone methyltransferase complex subunit ASH2(Human)
Memorial Sloan-Kettering Cancer Center

US Patent
LigandPNGBDBM685913(US12043645, Example 5)
Affinity DataIC50: 2.20E+3nMAssay Description:This assay relies on Whatman P-81 filter paper, which binds peptides but not SAM. Protein Methyl Transferases (PMTs) transfer 3H-Me of [3H-Me]-SAM to...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2024
Entry Details
US Patent