Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 12649
TargetBile acid receptor(Human)
CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang)

US Patent
LigandPNGBDBM50609047(CHEMBL5273113 | US12215098, Formula (I))
Affinity DataEC50:  13.8nMAssay Description:Purpose of the Assay:Activation of FXR binding reaction by the compound was detected by the amplified luminescent proximity homogeneous assay (alphas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2025
Entry Details
US Patent

TargetBile acid receptor(Human)
CSPC Zhongqi Pharmaceutical Technology (Shijiazhuang)

US Patent
LigandPNGBDBM50511109(Cilofexor | GS 9674 | Gs-9674 | PX-104 | PX104 | U...)
Affinity DataEC50:  65.2nMAssay Description:Purpose of the Assay:Activation of FXR binding reaction by the compound was detected by the amplified luminescent proximity homogeneous assay (alphas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2025
Entry Details
US Patent