Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 13118
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760334BDBM760334(1-(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- ...)
Affinity DataKi:  0.800nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760344BDBM760344(1-(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  1.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760333BDBM760333(1-(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- ...)
Affinity DataKi:  1.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605888BDBM50605888(CHEMBL5179759 | US12370182, Example 6)
Affinity DataKi:  2.70nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605882BDBM50605882(CHEMBL5202280 | US12370182, Example 1)
Affinity DataKi:  2.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605904BDBM50605904(CHEMBL5179688 | US12370182, Example 45)
Affinity DataKi:  3.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605868BDBM50605868(CHEMBL5186978 | US12370182, Example 8)
Affinity DataKi:  3.70nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605891BDBM50605891(CHEMBL5174560 | US12370182, Example 83)
Affinity DataKi:  3.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760297BDBM760297(4-(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- ...)
Affinity DataKi:  4.30nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760345BDBM760345(1-(4-fluorophenyl)-4-methyl- 5-({[6-(oxolane-2-car...)
Affinity DataKi:  4.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605890BDBM50605890(CHEMBL5200451 | US12370182, Example 3)
Affinity DataKi:  5nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605894BDBM50605894(CHEMBL5176630 | US12370182, Example 82)
Affinity DataKi:  5.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760338BDBM760338(2-fluoro-1-(2-{[1-(4- fluorophenyl)-4-methyl-1H- 1...)
Affinity DataKi:  5.30nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760346BDBM760346(1-(4-fluorophenyl)-4-methyl- 5-({[6-(oxolane-3-car...)
Affinity DataKi:  5.70nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605887BDBM50605887(CHEMBL5193778 | US12370182, Example 9)
Affinity DataKi:  6.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760370BDBM760370(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- yl]...)
Affinity DataKi:  6.5nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605886BDBM50605886(CHEMBL5197478 | US12370182, Example 7)
Affinity DataKi:  6.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605885BDBM50605885(CHEMBL5181374 | US12370182, Example 2)
Affinity DataKi:  7nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760331BDBM760331(cyclopropyl(2-{[1-(4- fluorophenyl)-4-methyl-1H- 1...)
Affinity DataKi:  7.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760352BDBM760352(1-(2-{[4-(4-chlorophenyl)-1- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  7.5nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605883BDBM50605883(CHEMBL5189320 | US12370182, Example 5)
Affinity DataKi:  7.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605892BDBM50605892(CHEMBL5178153 | US12370182, Example 84)
Affinity DataKi:  8.90nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760354BDBM760354(2-fluoro-1-(2-{[4-(4- fluorophenyl)-1-methyl-1H- 1...)
Affinity DataKi:  9.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760347BDBM760347(1-(4-fluorophenyl)-4-methyl- 5-({[6-(oxane-3-carbo...)
Affinity DataKi:  9.5nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760320BDBM760320(1-(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  9.80nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760295BDBM760295(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- yl]...)
Affinity DataKi:  11nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760337BDBM760337(2,2-difluoro-1-(2-{[1-(4- fluorophenyl)-4-methyl-1...)
Affinity DataKi:  11nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760339BDBM760339(1-(4-fluorophenyl)-4-methyl- 5-({[6-(oxane-4-carbo...)
Affinity DataKi:  13nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760326BDBM760326(1-(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  13nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760342BDBM760342(1-(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  13nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760296BDBM760296(2,2,2-trifluoro-1-(2-{[3-(4- fluorophenyl)-5-methy...)
Affinity DataKi:  14nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760317BDBM760317(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  14nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760341BDBM760341(5-[({6-cyclobutanecarbonyl- 5H,6H,7H-pyrrolo[3,4- ...)
Affinity DataKi:  14nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605884BDBM50605884(CHEMBL5193523 | US12370182, Example 4)
Affinity DataKi:  16nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760340BDBM760340(1-(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  17nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760313BDBM760313(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  18nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760357BDBM760357(4-(4-fluorophenyl)-1-methyl- 5-({[6-(oxolane-2-car...)
Affinity DataKi:  18nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760322BDBM760322(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  18nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760351BDBM760351(1-(2-{[4-(4-fluorophenyl)-1- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760294BDBM760294(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- yl]...)
Affinity DataKi:  21nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760316BDBM760316(2-{[1-(4-chlorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  22nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760323BDBM760323(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  24nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760304BDBM760304(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  24nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760348BDBM760348(4-(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  25nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760353BDBM760353(1-(2-{[4-(4-fluorophenyl)-1- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  25nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605901BDBM50605901(CHEMBL5207798 | US12370182, Example 14)
Affinity DataKi:  28nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760349BDBM760349(3-(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  28nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 50605898BDBM50605898(CHEMBL5184265 | US12370182, Example 78)
Affinity DataKi:  28nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760309BDBM760309(2-{[1-(4-fluorophenyl)-4- methyl-1H-1,2,3-triazol-...)
Affinity DataKi:  29nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 760356BDBM760356(1-(2-{[4-(4-fluorophenyl)-1- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  29nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/10/2025
Entry Details
US Patent

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