Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 13176
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765003BDBM765003(4-((1-(8-(6-(trifluoromethyl)pyridin-2-yl)-3,8-dia...)
Affinity DataIC50: 15nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764992BDBM764992(4-((1-(4-(5-(trifluoromethyl) pyrimidin-2-yl)piper...)
Affinity DataIC50: 18nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764986BDBM764986(4-((1-(4-(6-(trifluoromethyl) pyridin-2-yl)piperaz...)
Affinity DataIC50: 19nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764990BDBM764990(4-((1-(4-(6-methylpyridin-2- yl)piperazine-1-carbo...)
Affinity DataIC50: 23nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765004BDBM765004(4-((1-(5-(6-(trifluoromethyl)pyridin-2-yl)-2,5-dia...)
Affinity DataIC50: 26nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765025BDBM765025(4-((1-(4-(4-(trifluoromethyl)p yrimidin-2-yl)piper...)
Affinity DataIC50: 28nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764985BDBM764985(piperazine-1-carbonyl)cyclopentyl)amino)benzonitri...)
Affinity DataIC50: 32nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764986BDBM764986(4-((1-(4-(6-(trifluoromethyl) pyridin-2-yl)piperaz...)
Affinity DataIC50: 35nMAssay Description:Table 3.2: The cells were transferred to the perfusion tank and perfused with extracellular fluid. The intracellular fluid was: 130 mM K-aspartate; 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764981BDBM764981(4-((1-(4-(4-chloro-2-methoxy phenyl)piperazine-1-c...)
Affinity DataIC50: 35nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765022BDBM765022(piperazine-1-carbonyl)cyclopentyl)oxy)benzonitrile...)
Affinity DataIC50: 38nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764993BDBM764993(4-((1-(4-(4-(trifluoromethyl) pyrimidin-2-yl)piper...)
Affinity DataIC50: 38nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764970BDBM764970(4-((1-(4-(4-(trifluoromethyl)phenyl)piperazine-1-c...)
Affinity DataIC50: 40nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765032BDBM765032(4-((1-(4-(tert-butyl)piperazine- 1-carbonyl)cyclop...)
Affinity DataIC50: 51nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765053BDBM765053(2-(4-(tert-butyl)piperidine-1- carbonyl)-5-cyanoin...)
Affinity DataIC50: 53nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765005BDBM765005(4-((1-(4-(cyclopentanemethyl)piperazine-1-carbonyl...)
Affinity DataIC50: 54nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764970BDBM764970(4-((1-(4-(4-(trifluoromethyl)phenyl)piperazine-1-c...)
Affinity DataIC50: 56nMAssay Description:Table 3.2: The cells were transferred to the perfusion tank and perfused with extracellular fluid. The intracellular fluid was: 130 mM K-aspartate; 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764995BDBM764995(4-((1-(4-(6-(trifluoromethyl) pyridazin-3-yl)piper...)
Affinity DataIC50: 56nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764982BDBM764982(4-((1-(4-(3-methyl)phenyl)pi- perazine-1-carbonyl)...)
Affinity DataIC50: 64nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765023BDBM765023(4-((1-(4-(m-methylphenyl)pi perazine-1-carbonyl)cy...)
Affinity DataIC50: 65nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765025BDBM765025(4-((1-(4-(4-(trifluoromethyl)p yrimidin-2-yl)piper...)
Affinity DataIC50: 65nMAssay Description:Table 3.2: The cells were transferred to the perfusion tank and perfused with extracellular fluid. The intracellular fluid was: 130 mM K-aspartate; 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765055BDBM765055(2-(4-(tert-butyl)piperazine-1- carbonyl)-2,3-2H-5-...)
Affinity DataIC50: 68nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765020BDBM765020(4-((1-(4-(tert-butyl)piperidine- 1-carbonyl)cyclop...)
Affinity DataIC50: 72nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765029BDBM765029(4-((1-(8-(6-(trifluoromethyl) pyridin-2-yl)-3,8-di...)
Affinity DataIC50: 72nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765031BDBM765031(4-((1-(4-(tert-butyl)piperidine- 1-carbonyl)cyclop...)
Affinity DataIC50: 76nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765054BDBM765054(2-(4-(tert-butyl)piperidine-1- carbonyl)-2,3-2H-5-...)
Affinity DataIC50: 82nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765053BDBM765053(2-(4-(tert-butyl)piperidine-1- carbonyl)-5-cyanoin...)
Affinity DataIC50: 83nMAssay Description:Table 3.2: The cells were transferred to the perfusion tank and perfused with extracellular fluid. The intracellular fluid was: 130 mM K-aspartate; 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765010BDBM765010(4-((1-(4-(cyclohexyl)piperidine- 1-carbonyl)cyclop...)
Affinity DataIC50: 85nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764989BDBM764989(4-((3,3-dimethyl-1-oxo-1-(4- (6-trifluoromethyl)py...)
Affinity DataIC50: 87nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765006BDBM765006(4-((1-(4-(tert-butyl)piperidine-1-carbonyl)cyclope...)
Affinity DataIC50: 87nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764994BDBM764994(4-((1-(4-(6-(trifluoromethyl) pyridazin-3-yl)piper...)
Affinity DataIC50: 87nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765052BDBM765052(2-(4-(tert-butyl)piperazine-1- carbonyl)-5-cyanoin...)
Affinity DataIC50: 91nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765030BDBM765030(4-((1-(5-(6-(trifluoromethyl)p yridin-2-yl)-2,5-di...)
Affinity DataIC50: 91nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765018BDBM765018(4-((1-(4-(tert-butyl)piperidine- 1-carbonyl)tert-b...)
Affinity DataIC50: 91nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765008BDBM765008(4-((1-(4-(cyclopentyl)piperi dine-1-carbonyl)cyclo...)
Affinity DataIC50: 92nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765045BDBM765045(2-(4-(3-(trifluoromethyl)phe nyl)piperazine-1-carb...)
Affinity DataIC50: 92nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765006BDBM765006(4-((1-(4-(tert-butyl)piperidine-1-carbonyl)cyclope...)
Affinity DataIC50: 98nMAssay Description:Table 3.2: The cells were transferred to the perfusion tank and perfused with extracellular fluid. The intracellular fluid was: 130 mM K-aspartate; 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764971BDBM764971(4-((1-(4-(3-(trifluoromethyl) phenyl)piperazine-1-...)
Affinity DataIC50: 105nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765041BDBM765041(4-((1-(4-(tert-butyl)piperazine- 1-carbonyl)cyclop...)
Affinity DataIC50: 105nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765021BDBM765021(4-((1-(4-(tert-butyl)piperidine- 1-carbonyl)cyclop...)
Affinity DataIC50: 108nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765043BDBM765043(2-(4-(6-(trifluoromethyl)pyridin-2-yl)piperazine-1...)
Affinity DataIC50: 112nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765049BDBM765049(2-(4-(6-(trifluoromethyl)pyridin- 2-yl)piperazine-...)
Affinity DataIC50: 116nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764980BDBM764980(4-((1-(4-(4-(trifluoromethyl) phenyl)piperazine-1-...)
Affinity DataIC50: 129nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764979BDBM764979(4-((1-(4-(2-(trifluoromethoxy) phenyl)piperazine-1...)
Affinity DataIC50: 152nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765026BDBM765026(4-((1-(4-(4-(trifluoromethyl) pyrimidin-2-yl)piper...)
Affinity DataIC50: 182nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 764998BDBM764998(2-chloro-4-((1-(4-(6-(trifluoro methyl)pyridazin-3...)
Affinity DataIC50: 231nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765048BDBM765048(2-(4-(6-(trifluoromethyl)pyridin- 2-yl)piperazine...)
Affinity DataIC50: 261nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765019BDBM765019(4-((1-(4-(tert-butyl)piperidine- 1-carbonyl)cyclop...)
Affinity DataIC50: 280nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765050BDBM765050(2-(4-(6-methyl)pyridin-2-yl) piperazine-1-carbonyl...)
Affinity DataIC50: 285nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765009BDBM765009(4-((1-(8-aza-spiro[4.5]decane- 8-carbonyl)cyclopen...)
Affinity DataIC50: 287nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

TargetTransient receptor potential cation channel subfamily A member 1(Human)
Hangzhou Westan Pharmaceutical Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 765024BDBM765024(4-((1-(4-(trifluoromethyl)phe nyl)piperazine-1-car...)
Affinity DataIC50: 325nMAssay Description:Table 3.1: The cell analysis plate was placed in an FLIPR instrument (Molecular Probes), and the compound in the compound plate was added to the corr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/25/2025
Entry Details
US Patent

Displayed 1 to 50 (of 85 total ) | Next | Last >>
Jump to: