Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 13203
TargetMitogen-activated protein kinase 1(Human)
D3 Bio (Wuxi) Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 766787BDBM766787(US12398153, Compound WX003)
Affinity DataIC50: 0.290nMAssay Description:1. Purpose of the Assay:The ability of compounds to inhibit ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM MgCl2, 1 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Human)
D3 Bio (Wuxi) Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 766784BDBM766784(US12398153, Compound WX001A)
Affinity DataIC50: 0.310nMAssay Description:1. Purpose of the Assay:The ability of compounds to inhibit ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM MgCl2, 1 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Human)
D3 Bio (Wuxi) Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 766785BDBM766785(US12398153, Compound WX001B)
Affinity DataIC50: 0.320nMAssay Description:1. Purpose of the Assay:The ability of compounds to inhibit ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM MgCl2, 1 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Human)
D3 Bio (Wuxi) Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 766789BDBM766789(US12398153, Compound WX005)
Affinity DataIC50: 0.360nMAssay Description:1. Purpose of the Assay:The ability of compounds to inhibit ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM MgCl2, 1 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Human)
D3 Bio (Wuxi) Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 766786BDBM766786(US12398153, Compound WX002)
Affinity DataIC50: 0.400nMAssay Description:1. Purpose of the Assay:The ability of compounds to inhibit ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM MgCl2, 1 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Human)
D3 Bio (Wuxi) Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 766791BDBM766791(US12398153, Compound WX007)
Affinity DataIC50: 0.480nMAssay Description:1. Purpose of the Assay:The ability of compounds to inhibit ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM MgCl2, 1 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Human)
D3 Bio (Wuxi) Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 766790BDBM766790(US12398153, Compound WX006)
Affinity DataIC50: 0.940nMAssay Description:1. Purpose of the Assay:The ability of compounds to inhibit ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM MgCl2, 1 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent

TargetMitogen-activated protein kinase 1(Human)
D3 Bio (Wuxi) Co.

US Patent
LigandChemical structure of BindingDB Monomer ID 766788BDBM766788(US12398153, Compound WX004)
Affinity DataIC50: 1.10nMAssay Description:1. Purpose of the Assay:The ability of compounds to inhibit ERK2 kinase activity was measured.2. Assay Buffer:20 mM Hepes (pH 7.5), 10 mM MgCl2, 1 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/5/2025
Entry Details
US Patent