Report error Found 221 Enz. Inhib. hit(s) with all data for entry = 13248
Affinity DataIC50: 0.100nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.200nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.300nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.400nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.5nMAssay Description:Method (B): Measurement of A2a Binding Affinity Using SPABinding affinity using SPA was conducted as follows. Test compounds (50 nL) were dispensed i...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.5nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.5nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.600nMAssay Description:Method (B): Measurement of A2a Binding Affinity Using SPABinding affinity using SPA was conducted as follows. Test compounds (50 nL) were dispensed i...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.600nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.600nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.600nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.700nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.700nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.700nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.700nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 0.900nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.10nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.20nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.20nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.20nMAssay Description:The reported affinity of the compounds of the invention for the human A2b adenosine receptor was determined experimentally using a radioligand filtra...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.20nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.30nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.30nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.30nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.30nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.60nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.60nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 1.90nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.10nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.20nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.20nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.20nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.30nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.30nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.40nMAssay Description:The reported affinity of the compounds of the invention for the human A2b adenosine receptor was determined experimentally using a radioligand filtra...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.40nMAssay Description:Method (B): Measurement of A2a Binding Affinity Using SPABinding affinity using SPA was conducted as follows. Test compounds (50 nL) were dispensed i...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.5nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.60nMAssay Description:The reported affinity of the compounds of the invention for the human A2b adenosine receptor was determined experimentally using a radioligand filtra...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.70nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.70nMAssay Description:The reported affinity of the compounds of the invention for the human A2b adenosine receptor was determined experimentally using a radioligand filtra...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 2.90nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.20nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.60nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.60nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.10nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.20nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.40nMAssay Description:Method (A): Measurement of A2a Binding Affinity Using Radioligand Binding148 μL (5 μg/mL) membranes (Perkin Elmer, Cat. No. RBHA2aM400UA) and 2 μL co...More data for this Ligand-Target Pair
Ligand Info
