Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 1215
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39582BDBM39582(TJU-B183 | (Z)-N-(4-(benzo[d][1,3]dioxol-5-ylmethy...)
Affinity DataIC50: 100nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39582BDBM39582(TJU-B183 | (Z)-N-(4-(benzo[d][1,3]dioxol-5-ylmethy...)
Affinity DataIC50: 550nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39580BDBM39580(TJU-B182 | (Z)-5-(benzo[d][1,3]dioxol-5-ylmethylen...)
Affinity DataIC50: 550nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39580BDBM39580(TJU-B182 | (Z)-5-(benzo[d][1,3]dioxol-5-ylmethylen...)
Affinity DataIC50: 550nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 50594776BDBM50594776(CHEMBL5182235 | US12594261, Example 1)
Affinity DataIC50: 550nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 50594776BDBM50594776(CHEMBL5182235 | US12594261, Example 1)
Affinity DataIC50: 550nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39576BDBM39576(TJU-B076 | (Z)-5-(benzo[d][1,3]dioxol-5-ylmethylen...)
Affinity DataIC50: 5.50E+3nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39576BDBM39576(TJU-B076 | (Z)-5-(benzo[d][1,3]dioxol-5-ylmethylen...)
Affinity DataIC50: 5.50E+3nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39577BDBM39577(TJU-B116 | (Z)-5-(benzo[d][1,3]dioxol-5-ylmethylen...)
Affinity DataIC50: 5.50E+3nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetDual specificity protein kinase CLK1 [129-484](Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39577BDBM39577(TJU-B116 | (Z)-5-(benzo[d][1,3]dioxol-5-ylmethylen...)
Affinity DataIC50: 5.50E+3nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39576BDBM39576(TJU-B076 | (Z)-5-(benzo[d][1,3]dioxol-5-ylmethylen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39577BDBM39577(TJU-B116 | (Z)-5-(benzo[d][1,3]dioxol-5-ylmethylen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39580BDBM39580(TJU-B182 | (Z)-5-(benzo[d][1,3]dioxol-5-ylmethylen...)
Affinity DataIC50: 1.00E+4nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 50594776BDBM50594776(CHEMBL5182235 | US12594261, Example 1)
Affinity DataIC50: 1.00E+4nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Shanghai East Hospital

US Patent
LigandChemical structure of BindingDB Monomer ID 39582BDBM39582(TJU-B183 | (Z)-N-(4-(benzo[d][1,3]dioxol-5-ylmethy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Sanford-Burnham Center for Chemical Genomics (SBCCG) Sanford-Burnham Medical Research Institute (SBMRI, San Diego, CA) NIH Molecular Libraries Screen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2026
Entry Details
US Patent