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Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 13589
TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656032BDBM656032(2-fluoro-1-[6-({4-methyl-1-[6-(difluoromethyl)pyri...)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656030BDBM656030(1-[6-({1-[6-(difluoromethyl)pyridin-3-yl]-4-methyl...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656031BDBM656031(1-[6-({1-[6-(difluoromethyl)pyridin-3-yl]-4-methyl...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 655994BDBM655994(1-[6-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazo...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656014BDBM656014(2-fluoro-1-(3-{[5-methyl-3-(6-methylpyridin-3-yl)-...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656016BDBM656016(N-cyclopropyl-3-{[5-methyl-3-(6-methylpyridin-3-yl...)
Affinity DataKi:  2.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656009BDBM656009(1-(3-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazo...)
Affinity DataKi:  2.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 655997BDBM655997(2-methanesulfonyl-1-(6-{[5-methyl-3-(6-methylpyrid...)
Affinity DataKi:  3.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656015BDBM656015(2-methyl-1-(3-{[5-methyl-3-(6-methylpyridin-3-yl)-...)
Affinity DataKi:  4.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656012BDBM656012(5-{4-[({7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[...)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656006BDBM656006((5R)-1-methyl-5-(6-{[5-methyl-3-(6-methylpyridin-3...)
Affinity DataKi:  5.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656013BDBM656013(1-(3-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazo...)
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 655998BDBM655998(6-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazol-4...)
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656019BDBM656019(2-fluoro-1-(6-{[4-methyl-1-(6-methylpyridin-3-yl)-...)
Affinity DataKi:  6.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656008BDBM656008(1-ethyl-4-(6-{[5-methyl-3-(6-methylpyridin-3-yl)-1...)
Affinity DataKi:  6.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656002BDBM656002(6-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazol-4...)
Affinity DataKi:  7.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656018BDBM656018(1-(6-{[4-methyl-1-(6-methylpyridin-3-yl)-1H-1,2,3-...)
Affinity DataKi:  7.90nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656017BDBM656017(1-[3-({5-methyl-3-[6-(trifluoromethyl)pyridin-3-yl...)
Affinity DataKi:  8.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656003BDBM656003(1-methyl-4-(6-{[5-methyl-3-(6-methylpyridin-3-yl)-...)
Affinity DataKi:  8.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656005BDBM656005(1-methyl-5-(6-{[5-methyl-3-(6-methylpyridin-3-yl)-...)
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656037BDBM656037(2-fluoro-1-(6-{[1-methyl-4-(6-methylpyridin-3-yl)-...)
Affinity DataKi:  9.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656006BDBM656006((5R)-1-methyl-5-(6-{[5-methyl-3-(6-methylpyridin-3...)
Affinity DataKi:  9.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 655996BDBM655996(1-[6-({5-methyl-3-[6-(trifluoromethyl)pyridin-3-yl...)
Affinity DataKi:  9.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656011BDBM656011(2-methyl-5-[5-methyl-4-({[7-(oxane-4-carbonyl)-5H,...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656000BDBM656000(6-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazol-4...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656004BDBM656004(4-(6-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazo...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656010BDBM656010(4-(3-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazo...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656026BDBM656026(2-fluoro-1-[6-({4-methyl-1-[6-(trifluoromethyl)pyr...)
Affinity DataKi:  15nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 655999BDBM655999(4-(6-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazo...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656001BDBM656001(6-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazol-4...)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656022BDBM656022(1-(6-{[4-methyl-1-(6-methylpyridin-3-yl)-1H-1,2,3-...)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656033BDBM656033(1-(6-{[1-methyl-4-(6-methylpyridin-3-yl)-1H-1,2,3-...)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656023BDBM656023(2-cyclopropanecarbonyl-6-{[4-methyl-1-(6-methylpyr...)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656024BDBM656024(1-[6-({4-methyl-1-[6-(trifluoromethyl)pyridin-3-yl...)
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656020BDBM656020(2-methyl-1-(6-{[4-methyl-1-(6-methylpyridin-3-yl)-...)
Affinity DataKi:  30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656028BDBM656028(2-cyclopropanecarbonyl-6-({4-methyl-1-[6-(trifluor...)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656034BDBM656034(1-(6-{[1-methyl-4-(6-methylpyridin-3-yl)-1H-1,2,3-...)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656025BDBM656025(1-[6-({4-methyl-1-[6-(trifluoromethyl)pyridin-3-yl...)
Affinity DataKi:  33nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656038BDBM656038(1-(6-{[1-methyl-4-(6-methylpyridin-3-yl)-1H-1,2,3-...)
Affinity DataKi:  37.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 655995BDBM655995(tert-butyl 6-{[5-methyl-3-(6-methylpyridin-3-yl)-1...)
Affinity DataKi:  38nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656035BDBM656035(2-methyl-1-(6-{[1-methyl-4-(6-methylpyridin-3-yl)-...)
Affinity DataKi:  43nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656027BDBM656027(2-methyl-1-[6-({4-methyl-1-[6-(trifluoromethyl)pyr...)
Affinity DataKi:  44nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656021BDBM656021(3-methyl-1-(6-{[4-methyl-1-(6-methylpyridin-3-yl)-...)
Affinity DataKi:  48nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656036BDBM656036(2-cyclopropanecarbonyl-6-{[1-methyl-4-(6-methylpyr...)
Affinity DataKi:  52nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandChemical structure of BindingDB Monomer ID 656029BDBM656029(1-[3-({4-methyl-1-[6-(trifluoromethyl)pyridin-3-yl...)
Affinity DataKi:  99.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details US Patent