Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 11484
TargetE3 ubiquitin-protein ligase XIAP [241-356](Human)
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM620168(US20230295181, Compound 81)
Affinity DataKi:  55nMAssay Description:Compounds of the present disclosure were evaluated for potency and selectivity in a fluorescence polarization (FP) assay that measures inhibition of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [241-356](Human)
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM620169(US20230295181, Compound 82)
Affinity DataKi:  55nMAssay Description:Compounds of the present disclosure were evaluated for potency and selectivity in a fluorescence polarization (FP) assay that measures inhibition of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [241-356](Human)
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM391840(US10300074, Compd 35 | US20230295181, Compound A)
Affinity DataKi:  55nMAssay Description:Compounds of the present disclosure were evaluated for potency and selectivity in a fluorescence polarization (FP) assay that measures inhibition of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [241-356](Human)
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM620153(US20230295181, Compound 65)
Affinity DataKi:  55nMAssay Description:Compounds of the present disclosure were evaluated for potency and selectivity in a fluorescence polarization (FP) assay that measures inhibition of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [241-356](Human)
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM620165(US20230295181, Compound 80)
Affinity DataKi:  55nMAssay Description:Compounds of the present disclosure were evaluated for potency and selectivity in a fluorescence polarization (FP) assay that measures inhibition of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [241-356](Human)
Sanford Burnham Prebys Medical Discovery Institute

US Patent
LigandPNGBDBM620148(US20230295181, Compound 38)
Affinity DataKi:  66nMAssay Description:Compounds of the present disclosure were evaluated for potency and selectivity in a fluorescence polarization (FP) assay that measures inhibition of ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent